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4-(2-phenylpyrrolidine-1-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
1-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperidine-3-carboxamide
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[1-(5-chloro-2-methylbenzoyl)pyrrolidin-3-yl]benzoic acid
2-amino-6-(4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}piperazin-1-yl)pyrimidin-4-ol
2-methyl-8-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-2,8-diazaspiro[4.5]decan-3-one
N-[3-({[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-2-(2-methoxy-5-methylphenyl)acetic acid
N-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]-4-fluorobenzamide
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-2-amine
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-[(3-hydroxyazetidin-1-yl)methyl]piperidin-2-one
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2-(2-methoxyethyl)piperidine
methyl 3-[(2-methyl-1H-indol-3-yl)methyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
1-[2-(3-methoxyphenoxy)ethyl]-4-(1H-pyrazole-3-carbonyl)piperazine
1-[2-(4,4-difluoropiperidin-1-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
(3R,5S)-N3-[(1-ethyl-1H-imidazol-2-yl)methyl]-N3-methyl-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
(4aS,8aR)-1-(2-hydroxyethyl)-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-cyclobutyl-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-({[(3-hydroxypyrrolidin-3-yl)methyl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethan-1-one
3-{[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
6-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
N-[1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4S)-3-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-4-(propan-2-yl)-1,3-oxazolidin-2-one
(2S,4S)-4-amino-1-[4-methoxy-3-(methoxymethyl)benzoyl]-N-methylpyrrolidine-2-carboxamide
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2,3-dihydro-1,4-benzodioxine-5-carboxamide
3-hydroxy-S-[2-(2-methoxyacetyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
3-{2-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
1-[1-(4-methyl-1H-pyrrole-2-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-3-azaspiro[5.5]undecan-9-amine
7-[(3-methoxyphenyl)methyl]-2-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-[(3-chlorophenyl)methyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
4-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}-N-propylaniline
3-amino-1-{[1-(pyridin-4-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-3-carboxylic acid
1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(dimethylamino)-N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-{furo[3,2-c]pyridin-4-yl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3S,4R)-1-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-3-methoxypiperidin-4-amine
(3S,4S)-1-(9H-purin-6-yl)piperidine-3,4-diol
[(3-chlorophenyl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine