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N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
5-hydroxy-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-[(4-methoxypyridin-2-yl)methyl]benzamide
(2-{1-[4-(2-methoxyphenyl)benzoyl]piperidin-2-yl}ethyl)dimethylamine
8-fluoro-3-[2-(piperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-(3-hydroxy-3-methylbutyl)-N-(3-methoxypropyl)-N-methylbenzamide
3-cyclopentyl-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-(2-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-7-yl)-2,2-dimethylpropan-1-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[1-(2-chlorophenyl)cyclopropyl]-2-(methylamino)pyridine-4-carboxamide
6-(4-fluorophenyl)-7-methyl-8-oxo-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1R,2S,6R,7S)-4-[2-(1H-imidazol-2-yl)benzoyl]-4-azatricyclo[5.2.2.02,6]undecane
2-(3-hydroxypropyl)-8-[2-(2-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(3-methylbut-2-en-1-yl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-[(4-chlorophenyl)methyl]-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1,3-benzoxazole-5-carboxamide
3-[(4-methylpiperazin-1-yl)sulfonyl]-N-(oxolan-2-ylmethyl)-5-phenylbenzamide
1-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-3-(dimethylamino)propan-2-ol
N-(2,3-dihydroxypropyl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N4-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N,N,3-trimethyl-4-({[(1-propyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)benzamide
5-phenyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-(3-chlorophenyl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-[methyl(piperidin-4-yl)amino]ethan-1-one
N-ethyl-2-{4-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]piperazin-1-yl}acetamide
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
2-[3-(2-methoxyethyl)-5-[4-(5-methylfuran-2-yl)phenyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
1-[(3-fluorophenyl)methyl]-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
N-(4-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}-4-oxobutyl)acetamide
N-[2-(4-chlorophenyl)ethyl]-4-cyano-1-methyl-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide
5-(5-chlorothiophen-2-yl)-1-cyclohexyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
(1S,5R)-6-benzyl-3-[(3-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
2-(4-{2-[(4-chlorophenyl)methyl]-1,3-benzoxazole-5-carbonyl}piperazin-1-yl)phenol
1-{5-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-2-methylphenyl}imidazolidin-2-one
2-(2,3-dimethylphenoxy)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1,4-dimethyl 2-[(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}phenyl)formamido]butanedioate
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-[(2-methylphenyl)methyl]acetamide
N-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 4-{2-amino-6-oxo-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl}-1H-pyrazole-3-carboxylate
{1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
methyl 3-[2-(cyclohex-1-en-1-yl)acetyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
N-[2-(4-methoxyphenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(2S,4S)-N-[(2-fluorophenyl)methyl]-4-(2-methoxyacetamido)-1-methylpyrrolidine-2-carboxamide