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7-(2-hydroxyethyl)-2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(6-methylpyridin-2-yl)ethyl]acetamide
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-(4-methyl-1H-pyrazol-3-yl)piperidine
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl][2-methyl-2-(morpholin-4-yl)propyl]amine
(1R,5S,8S)-N-(6-chloropyridin-3-yl)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
5-butyl-1'-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
5-[(isoquinolin-5-yloxy)methyl]-N-[(2S)-oxolan-2-ylmethyl]-1,2-oxazole-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-N,2-dimethyl-6-propylpyrimidin-4-amine
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-methylphenoxy)ethyl]acetamide
2-cyclopentyl-N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
4-(2-chloro-6-fluoro-3-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-ethyl-4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1-methylpiperazin-2-one
ethyl 4-{4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}piperidine-1-carboxylate
(2S)-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carboxylic acid
7-fluoro-2-methyl-N-[2-(pyridin-3-yl)ethyl]quinoline-4-carboxamide
2-(3,5-difluorophenyl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-3-methylpiperidine
2-ethoxy-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[2-(3-methoxyphenyl)ethyl]piperidine
6-(aminomethyl)-N-[2-(4-chlorophenyl)-2-(piperidin-1-yl)ethyl]-2-methylpyrimidin-4-amine
N-[(3-chlorophenyl)methyl]-1-methyl-3-(propan-2-yl)-N-propyl-1H-pyrazole-5-carboxamide
3-methyl-6-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyridazine
2-cyclopentyl-N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-acetyl-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}piperidine-4-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-(1-methylpiperidin-2-yl)propanamide
1-(carbamoylmethyl)-N-[3-(1H-indazol-1-yl)propyl]piperidine-4-carboxamide
{2-[4-(4-cyanophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}urea
1-cyclopropanecarbonyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]piperidine-4-carboxamide
2-cyclopropyl-N-({1-[(4-hydroxyquinolin-2-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
1-[(diethylcarbamoyl)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
1-{2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]phenyl}-1,3-diazinane-2,4-dione
1-[(3-fluorophenyl)methyl]-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
2-(4-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}morpholin-3-yl)acetic acid
3-(1,2-oxazolidin-2-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
(2S,4R)-1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-1,3-benzothiazole
1-{1-[6-(aminomethyl)pyrimidin-4-yl]piperidin-4-yl}-3-phenylpropan-1-ol
[1-(2-aminopyrimidin-4-yl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
4-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
5-benzyl-N-methyl-N-(oxan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2S,4R)-N,N-diethyl-4-[3-(4-hydroxyphenyl)propanamido]-1-methylpyrrolidine-2-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
(4aS,8aR)-6-(5-chloropyrimidin-2-yl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(pyrazin-2-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide