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2-(3-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}phenyl)ethan-1-amine
ethyl 3-[(2-methylphenyl)methyl]-1-(2-oxo-2-phenylacetyl)piperidine-3-carboxylate
(3R,4S)-4-(5-methylfuran-2-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidin-3-amine
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}pyridine
4-[(4-chlorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-phenyl-1-[1-(5-phenyl-1,2,4-triazin-3-yl)piperidin-4-yl]ethan-1-ol
4-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)-3-(2-hydroxyethyl)piperazin-2-one
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-yl)propanamide
5-[3-(morpholin-4-ylmethyl)phenyl]pyridine-3-carboxamide
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-6-methoxy-3,4-dihydroquinazolin-4-one
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-2-one
6-ethyl-2-methyl-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(1-phenylcyclopropyl)azepan-4-amine
2-benzyl-1-methyl-N-[(3S)-2-oxoazepan-3-yl]-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-N-[(2-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
{2-[4-(2,3-dihydro-1-benzofuran-7-carbonyl)morpholin-2-yl]ethyl}dimethylamine
7-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
(2R,3R,6R)-3-phenyl-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(2,1,3-benzothiadiazol-5-yl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-(3-phenylpropyl)-4-(thian-4-yl)morpholine
4-cyclopropyl-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-methylpyrrolidin-2-one
(2,1,3-benzothiadiazol-5-ylmethyl)[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]methylamine
(3aS,6aS)-5-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 1-[2-(ethylsulfanyl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(5-methylfuran-2-yl)ethyl]amino}methyl)piperidin-2-one
N1-(3-methylpyridin-4-yl)-N2-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}ethane-1,2-diamine
N-(3-chloro-4-propanamidophenyl)-2-methoxypyridine-4-carboxamide
2-{2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethoxy}acetamide
6-(2-aminoethyl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
N,N-dimethyl-2-{[(5-methylthiophen-2-yl)formamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-ethyl-N,2,5-trimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrrole-3-carboxamide
(4aS,8aR)-N-(furan-2-ylmethyl)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
(2S,4S)-4-cyclopropaneamido-N-ethyl-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidine-2-carboxamide
{1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-yl}methanol
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-[2-(4-propanoylphenyl)ethyl]-1λ6-thiolane-1,1-dione
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
(3aS,6aS)-2-ethyl-5-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-methyl-1,3-benzoxazol-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(methoxymethyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
3-{2-[4-(2-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
3-[2-(piperidin-2-yl)ethyl]-5-(quinolin-8-yl)phenol
(3S,4S)-1-(4-amino-5-methylpyrimidin-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-(1-phenylethyl)-3-{[2-(pyridin-2-yl)ethyl]amino}propanamide