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(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(3,4-difluorophenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
5-[(2S)-1-cyclohexanecarbonylpyrrolidin-2-yl]-1-methyl-1H-1,2,4-triazole
3-[(1-benzofuran-2-ylmethyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrazin-2-amine
2-[1-(1-methylpiperidin-4-yl)-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
6-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
(1S,4R)-1-({[9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]sulfonyl}methyl)-7,7-dimethylbicyclo[2.2.1]heptan-2-one
4-methyl-3-[5-(1-methylpiperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
4-fluoro-N-(3-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-oxopropyl)benzamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-3-(4-ethylphenyl)propan-1-one
(1R,3S)-3-ethoxy-7-[2-(methylamino)pyridine-4-carbonyl]-7-azaspiro[3.5]nonan-1-ol
2-[1-(3-phenylpropyl)-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
6-chloro-N-(1-methylpiperidin-4-yl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
2-(propylsulfanyl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-{4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-N-methylpyridine-3-carboxamide
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(2-phenylethyl)acetamide
N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-4-(5-chloropyridin-2-yl)piperazine-1-carboxamide
{5-chloro-7-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-methyl-5-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}-3,4-dihydropyrimidin-4-one
N-methyl-2-(3-oxo-1-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-2-yl)acetamide
3-(N-methyl-1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
1-(4-methoxyphenyl)-3-methyl-4-[3-(pyridin-2-yl)propanoyl]piperazin-2-one
7-(2-cyclohexylethyl)-2-(2-methoxypyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decane
4-{6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}-2-methoxypyridine-3-carbonitrile
1-(2-{[(4-acetamidophenyl)methyl]amino}ethyl)-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-cyclopropyl-1-(4-phenoxybutanoyl)pyrrolidine-3-carboxylic acid
3-[(2,5-dimethoxyphenyl)methyl]-3H,4H-pyrido[2,3-d]pyrimidin-4-one
{4-[(2-chlorophenyl)methyl]-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl}methanol
(5-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}furan-2-yl)methanol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]ethan-1-one
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-S-(4-fluoro-2-methylphenyl)-2-oxoethane-1-sulfonamido
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]pyrimidin-2-amine
2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxylic acid
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(phenylamino)pyrimidine-5-carboxamide
4-(2-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}-2-methylpropyl)morpholine
dimethyl(1-{3-[4-(morpholin-4-yl)phenyl]phenyl}ethyl)amine
4-(2,2-dimethylpropanoyl)-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidine
methyl 3-(cyclobutylmethoxy)-5-{[(2S)-1-hydroxypropan-2-yl]carbamoyl}benzoate
{4-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}methanol
N-cyclopropyl-1-{1-[(2-fluoro-3-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
6-(aminomethyl)-2-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidin-4-amine
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(morpholin-4-yl)ethyl]acetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-4-(1H-pyrazol-5-yl)benzamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
methyl (2S,4R)-4-(dimethylamino)-1-[2-(1-methyl-1H-indol-3-yl)acetyl]pyrrolidine-2-carboxylate