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N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
5-(4-methoxyphenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carbonitrile
2-(2-aminoethyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]quinazolin-4-amine
5-[3-(benzyloxy)piperidine-1-carbonyl]-2-ethylpyrimidine
N-[2-(methylsulfanyl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
N-methyl-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
ethyl 4-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]-1H-pyrazole-3-carboxylate
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-(5-methyl-2H-1,2,3-triazole-4-carbonyl)piperidin-3-yl]methanol
1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)-N-[(5-methylfuran-2-yl)methyl]propanamide
4,6-dimethoxy-2-[4-(1-methyl-1H-1,2,4-triazol-5-yl)phenyl]pyrimidine
3-(morpholine-4-sulfonyl)-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzoic acid
1-(cyclohexylmethyl)-5-(4-hydroxypiperidin-1-yl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-2-[methyl(pyridin-2-ylmethyl)amino]-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
(5S,9aS,9bS)-5-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanoic acid
3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)azepan-2-one
3-methanesulfonyl-N-[(3R,4S)-1-(2-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]propanamide
N-(2,6-dimethylphenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
2-(3-methylbutyl)-8-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
6-(2-aminoethyl)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N,2-dimethylpyrimidin-4-amine
3-(carbamoylmethoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
2-[1-(2-methylpropyl)-4-phenyl-1H-imidazol-5-yl]-1,3-thiazole
5-ethyl-4-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]pyrimidin-2-amine
1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-phenylpiperidine-4-carbonitrile
5-propyl-1'-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-4-methylbenzamide
(4aS,8aR)-6-(furan-2-carbonyl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{[(cyclopropylmethyl)(propyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-cyclopropyl-N-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-2-phenylethyl}pyridine-2-carboxamide
2-amino-6-[4-fluoro-2-(trifluoromethyl)phenyl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-3-(3-methylphenyl)piperidine
2-{4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]-2,6-dimethoxyphenoxy}propanoic acid
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]acetamide
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
7-chloro-2-(furan-2-yl)-N,8-dimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]quinoline-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(3-methoxyphenyl)methyl]-N-methylbenzamide
3-chloro-4-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
1-benzoyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidin-4-amine
2-[5-(3,5-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]-2-methylpropane-1,3-diol
2-methyl-6-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
N-butyl-4-hydroxy-2-(4-methylphenyl)-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
5-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]pyridine-2,4-diol