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N5-cyclooctyl-N3-(furan-2-ylmethyl)-N3-methyl-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-4-(3-fluorophenyl)-1-(2-methanesulfonylethyl)pyrrolidine-3-carboxylic acid
3-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-6-methylquinolin-2-ol
1-[4-(1-carbamoyl-1-methylethyl)phenyl]-3-phenyl-1H-pyrazole-4-carboxylic acid
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
4-{[1-(3-fluorophenyl)-5-[(2-methoxyethoxy)methyl]-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
N-(1-benzylpiperidin-4-yl)-2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-6-(2-methoxyphenyl)pyridine-3-carboxamide
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzenesulfonamide
2-(1,4-oxazepan-4-ylmethyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidine-2-carboxamide
2-(3,5-dimethyl-4-phenyl-1H-pyrazol-1-yl)-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[(3-methylquinoxalin-2-yl)methyl]piperidine-4-carboxylic acid
1-(piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
5-{[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}quinoxaline
2-(4-fluorophenyl)-N-[2-(pyridin-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-(4-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}phenoxy)acetic acid
methyl (2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}pyrrolidine-2-carboxylate
1-methyl-5-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]-1,2-dihydropyridin-2-one
3-(propan-2-yl)-5-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
1-[2-(dimethylamino)-4-{[(2,5-dimethylphenyl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-5,6-dimethylpyridine-3-carbonitrile
8-[(5-ethylpyridin-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-2-methyl-2,3-dihydropyridazin-3-one
3-[(3R,4S)-1-(isoquinolin-1-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylbenzamide
1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}azepan-4-amine
2-amino-1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
[5-(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
(2S,4R)-4-amino-1-[2-(2,5-dimethoxyphenyl)acetyl]-N-ethylpyrrolidine-2-carboxamide
2-({4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}sulfanyl)ethan-1-ol
1-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-methyl-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
2-[2-(3-fluorophenyl)ethyl]-6,7-dimethoxyquinazolin-4-amine
(3aR,7aS)-2-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(4S)-3-{2-oxo-2-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-4-phenyl-1,3-oxazolidin-2-one
4-{4-[3-(2-fluorophenoxy)azetidin-1-yl]piperidin-1-yl}-2-methyl-6-propylpyrimidine
3-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
5-({[1-(dimethylcarbamoyl)piperidin-3-yl]formamido}methyl)thiophene-2-carboxylic acid
4-{5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-pyrazol-3-yl}phenol
1-[(1S,5R)-6-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]pyridin-3-amine
(3S,4S)-1-(1-benzothiophen-3-ylmethyl)-4-methylpiperidine-3,4-diol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
5-[5-(1H-1,3-benzodiazol-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-N-ethylpyrimidin-2-amine
methyl[(3-methyl-1H-indol-2-yl)methyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
(4aS,7aR)-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidine-4-carboxamide
(4aS,8aR)-6-(2,6-dimethylpyrimidine-4-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-[(4-cyclopentylpiperazin-1-yl)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one