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N-methyl-4-[2-oxo-2-(piperidin-1-yl)ethoxy]-N-[1-(pyridin-3-yl)ethyl]benzamide
1-(2-chlorophenyl)-3-{1-[1-(oxolane-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
4-{1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}pyridine
3-chloro-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyridine-4-carboxamide
2-{4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-4-carbonitrile
1-methyl-9-(2-methyl-5-propylpyrimidin-4-yl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-(3-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
methyl 2-({[4-(cyclobutylmethoxy)phenyl]methyl}(cyclopropyl)sulfamoyl)benzoate
3-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
1-[4-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)phenyl]ethan-1-one
N-ethyl-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidine-3-carboxamide
N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(trifluoromethyl)pyrimidin-4-amine
5-[3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)propyl]-1,3,4-thiadiazol-2-amine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2,3-dihydro-1-benzofuran-5-carboxamide
5-methyl-2-(4-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidin-4-amine
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-(2-methoxyphenyl)-4-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]piperazine
1-[(1-phenylcyclopentyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
1-[(3,4-dimethylphenyl)methyl]-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-2-one
2-[2-(dimethylamino)-2-(3-methylphenyl)-N-(1-methylpiperidin-4-yl)acetamido]acetic acid
N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
1-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
4-fluoro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-cyclopropyl-3-(4-methoxyphenyl)-3-(2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione
N-[(3S,4R)-1-(2,6-dimethylbenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}-6-(propan-2-yl)pyridine-3-carbonitrile
4-[(1,4-dimethylpiperidin-4-yl)methyl]-1-(2-phenylethyl)piperazin-2-one
2-[2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)ethyl]-1,3-thiazole-4-carboxylic acid
N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
2-(2-chloro-6-fluorophenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(2-methylpropyl)-8-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
5-{1-[2-(propane-2-sulfonyl)ethyl]-1H-imidazol-2-yl}quinoline
1-(butan-2-yl)-5-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethyl)-1H-indole
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[(furan-2-ylmethyl)(methyl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
4-benzoyl-N-benzylpiperidine-1-sulfonamide
(4S)-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
(3S,4S)-1-[(9-ethyl-9H-carbazol-3-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
7-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(4aS,8aR)-6-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
1-[2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-2-oxoethyl]-3,3-dimethylurea
3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3H,4H-pyrido[4,3-d]pyrimidin-4-one
1-methyl-1'-(5-phenyl-1,2-oxazole-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one