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1-methyl-9-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
2-(dimethyl-1,2-oxazol-4-yl)-3-methylquinoxaline
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]thiophene-3-sulfonamide
2-{2-[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,3-benzothiazole
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
1-(3-methoxyphenyl)-6-methyl-4-[2-(4-methylphenoxy)acetyl]piperazin-2-one
N-(3-{4-[benzyl(2-hydroxyethyl)amino]piperidin-1-yl}phenyl)-4-fluorobenzene-1-sulfonamide
(4aS,7aR)-6,6-dioxo-N-(propan-2-yl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
8-{2-[cyclopentyl(methyl)amino]acetyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2,3-dimethylphenyl)methyl]-2-(1-methylpiperidin-2-yl)acetamide
6-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-4-methylpiperazine
1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
3-(2-methylphenyl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N5-cyclobutyl-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-(methoxymethyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}furan-2-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(1,3-thiazol-2-ylmethyl)pyrimidin-2-amine
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-N-(2,2,2-trifluoroethyl)-1,4-dihydropyridine-3-carboxamide
1-(2,5-dimethylphenyl)-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-3-phenyl-1H-pyrazole
N-cyclooctyl-3-{[3-(1H-imidazol-1-yl)propyl]amino}propanamide
6-(methoxymethyl)-1-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2E)-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(furan-2-yl)prop-2-en-1-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(5-propylfuran-2-yl)methyl]amine
4-(2-fluorophenoxy)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
N-methyl-4-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)pyridin-2-amine
5-fluoro-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1H-indole-2-carboxamide
2-[2-(2-methylpyrrolidin-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indazol-3-one
6-[(3S)-3-ethylmorpholine-4-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-ethyl-9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(2-methoxyethyl)-3-[4-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(2-fluorophenyl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(2-chlorophenyl)-1-(4-fluorophenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
3-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
[3-({1-[2-(pyrrolidin-1-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
N-[(3-methoxyphenyl)methyl]-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-(prop-2-en-1-yl)benzamide
2-[2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]-6-methyl-3,4-dihydropyrimidin-4-one
N-(1-hydroxybutan-2-yl)-2-[(prop-2-en-1-yl)amino]benzamide
8-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(1,2-oxazolidin-2-yl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridine
1-(4-fluorophenyl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]cyclopropane-1-carboxamide
4-(3,3-diphenylpiperidin-1-yl)butanamide
4-(benzenesulfonyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
4-(4-oxo-7-{[(propan-2-yl)carbamoyl]carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
N-methyl-N-{2-phenyl-1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]ethyl}thiophene-3-carboxamide