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1-(1-methyl-1H-pyrrol-2-yl)-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethane-1,2-dione
N'-cyclopentyl-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)butanediamide
N-(1-cycloheptylpiperidin-3-yl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
3-[(2-chlorophenyl)methyl]-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(5-methanesulfonyl-2-methylphenyl)-4-phenylazepane-1-carboxamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-({[(2S)-2-aminopropyl]amino}methyl)-6-fluoroquinolin-4-ol
3-cyclopropyl-6-{pyrazolo[1,5-a]pyrimidin-3-yl}-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-({1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)-1-(pyrrolidin-1-yl)ethan-1-one
1-methyl-4-[2-(3,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]piperidine
2-amino-N,N-dimethyl-4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-sulfonamide
4-(4-{8-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenyl)-2-methylbut-3-yn-2-ol
ethyl 4-[4-oxo-2-(propan-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-8-yl]piperidine-1-carboxylate
4-(2-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}ethyl)morpholine
N2-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
(3S,5R)-N5-(4-fluorophenyl)-N3,N3-dimethyl-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
1,8-bis(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-3-[methyl({[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl})amino]propanamide
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
5-(2-phenoxyphenyl)furan-2-carboxamide
6-fluoro-2-({[3-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)quinolin-4-ol
1-{3-oxo-3-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-(quinoxalin-2-ylmethyl)acetamide
N-[(2-fluorophenyl)methyl]-2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]acetamide
6-[2,4-dichloro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
methyl 2-(cyclopropylsulfamoyl)-6-(3,4-dimethylbenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-4-(6-methyl-2-propylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]methyl}benzonitrile
1-(carbamoylmethyl)-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-(pyrrolidin-1-yl)pentanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
6-(2-aminoethyl)-N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-methylpyrimidin-4-amine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
2-{[3-(furan-2-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-(2-{1-[(2R)-2-amino-3-phenylpropanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2-(morpholin-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
7-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
7-[(3-hydroxybutyl)sulfamoyl]-N-propyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
N-cyclopropyl-N-[(3-methoxyphenyl)methyl]-2-(morpholin-2-yl)acetamide
N-{2-[(2,6-dimethylphenyl)carbamoyl]phenyl}pyridine-3-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-(pyridine-3-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-{3-[(2,2-dimethylpyrrolidin-1-yl)methyl]phenoxy}-2-hydroxypropyl)piperidin-4-ol
2-(azepan-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
N-(cyclopent-3-en-1-yl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-(2-oxopyrrolidin-1-yl)butanamide
N-({5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide