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(3S,4R)-1-[2-(2,4-difluorophenyl)acetyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
6-fluoro-4-[2-(3-methoxypropyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
3-{5-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]thiophen-2-yl}prop-2-yn-1-ol
4-{methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-1,2,5-thiadiazole-3-carboxamide
N-ethyl-6-[(2-phenoxyethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(1-methyl-1H-indol-6-yl)methyl]amine
5-[1-(difluoromethyl)-5-methyl-1H-pyrazol-4-yl]-8-methoxyquinoline
1-(2-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
8-(1-ethyl-1H-pyrazole-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-ethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
N-[(1-methyl-1H-indol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-[2-(azepan-1-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-(propan-2-yl)acetamide
4-chloro-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1H-pyrazol-5-amine
4-[5-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)pyrimidin-2-yl]morpholine
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl](4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
4-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
2-{2-[2-(1H-imidazol-2-yl)benzoyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
N-[2-(1H-pyrazol-1-yl)ethyl]-1-benzofuran-5-carboxamide
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(pyrimidin-2-yloxy)phenyl]methyl})amine
2,6-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]quinoline-3-carboxamide
N'-(2-ethoxyphenyl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}propanediamide
3-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
(1R,3S)-7-{[3-(4-chlorophenoxy)phenyl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
5-cyclopropyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,3-oxazole-4-carboxamide
5-[(3-ethoxypropyl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(cyclopent-1-ene-1-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
(3aS,7aR)-2-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-hydroxy-N-[1-(pyrazin-2-yl)propan-2-yl]pyridine-4-carboxamide
2-methyl-6-(1-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)pyrimidin-4-ol
3-(azepane-1-carbonyl)-N-[(2,3-dimethoxyphenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-cyclopropyl-N-(1,4-dioxan-2-ylmethyl)-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
2-{5-[1-(3-methylphenyl)-1H-imidazol-2-yl]-4-phenyl-1H-imidazol-1-yl}ethan-1-ol
N-cyclopropyl-3-pentanamido-N-(1,3-thiazol-5-ylmethyl)benzamide
3-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
3-methyl-8-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
4-cyclobutanecarbonyl-N-(4-phenylphenyl)-1,4-diazepane-1-carboxamide
N-[2-(1-ethylpiperidin-3-yl)ethyl]-4-hydroxy-3-methylbenzamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-(2-hydroxy-2-phenylethyl)-1,2-oxazole-3-carboxamide
N-(2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}ethyl)-N-methylmethanesulfonamide
4-({2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)-2-ethoxyphenol
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-[3-(pyridin-2-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(1r,4r)-N-benzyl-4-hydroxy-N-[(3-methylpyridin-2-yl)methyl]cyclohexane-1-carboxamide
1-{3-[2-(methoxymethyl)piperidine-1-carbonyl]benzenesulfonyl}azetidin-3-ol
methyl 2-(diethylsulfamoyl)-6-(1-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate