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{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[1-(dimethylamino)propan-2-yl]amine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(6-phenoxypyridin-3-yl)-1-[(trimethylpyrazin-2-yl)methyl]piperidine-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-benzofuran-2-ylmethyl)-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
2-methyl-6-{1-[(5-phenylthiophen-2-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
(3S,4R)-1-cyclopentanecarbonyl-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(2-chloro-6-fluorophenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
5-ethyl-1'-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(4-cyclohexylpiperazin-1-yl)methyl]-4-(2,5-dimethoxyphenyl)phenol
2-{1-[(4-methylphenyl)methyl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[1-(thiophen-2-yl)propyl]piperidine-4-carboxamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-amino-N-[2-(2-chlorophenyl)ethyl]-4-phenylpyrimidine-5-carboxamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-(oxan-4-yl)benzamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(2-methylbutyl)piperidine
1-[2-(2-phenylazetidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
3-[(2-fluorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
N-benzyl-1-[1-(2-cyclopropylacetyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(1S,5R)-3-(3-chlorothiophene-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2,3-dimethoxybenzamide
N-benzyl-3-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,2-oxazole-5-carboxamide
(2S)-N2-ethyl-N1-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1,2-dicarboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl 2-{[2-(4-carbamoylphenyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}acetate
1-(2-ethoxyethyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(piperidin-1-yl)piperidine-4-carboxamide
N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-(1-phenylpiperidin-4-yl)-4-(piperidin-1-yl)butanamide
3-chloro-1-[2-(6-hydroxy-1,4-oxazepan-4-yl)-2-oxoethyl]-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl][(2,3-difluoro-4-methylphenyl)methyl]methylamine
N-(butan-2-yl)-3-(methylsulfanyl)-N-(pyridin-3-ylmethyl)propanamide
2-methoxy-6-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]acetamide
8-[2-(methylsulfanyl)propanoyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
3-(prop-2-en-1-yl)-1-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
4-(1H-1,3-benzodiazole-5-carbonyl)-3-butyl-1-methylpiperazin-2-one
1-[(3-ethoxy-4-methoxyphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
4-benzyl-1-[(6-chloropyridin-2-yl)methyl]-3-ethyl-1,4-diazepan-5-one
8-fluoro-2-[2-(1H-imidazol-4-ylmethyl)-3-oxopiperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-(oxan-4-yl)-N-(2-phenoxyethyl)piperidine-3-carboxamide
N-{4-[2-(3,5-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]phenyl}acetamide
N-cyclopropyl-1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-methoxy-N-{1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
3-{11-methyl-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-4-yl}propanamide