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N4-(2-ethoxypropyl)-5-ethyl-N4,6-dimethylpyrimidine-2,4-diamine
1-[7-(cyclohex-3-en-1-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-4-ol
1-(6-cyanopyridin-2-yl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
N-cyclopropyl-3-({1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
[(2S)-1-{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}pyrrolidin-2-yl]methanol
(4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,4-oxazepan-6-yl)methanol
N-methyl-N-(1-methylpyrrolidin-3-yl)-4-propylpyrimidine-5-carboxamide
2-[5-(methoxymethyl)furan-2-carbonyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(2-{3-[3-(3,6-dimethylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)dimethylamine
(2S,4S)-4-amino-1-methyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrrolidine-2-carboxamide
methyl 2-{[(3,4-difluorophenyl)methyl]sulfamoyl}-6-(2,2-dimethylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N,3-dimethyl-4-[({2-[(trifluoromethyl)sulfanyl]ethyl}carbamoyl)amino]benzamide
(4aS,7aR)-1-[2-(2-chlorophenoxy)acetyl]-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-(5-propyl-1,2-oxazole-3-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
1-{2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyrrolidin-2-one
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-phenoxypropanamide
ethyl 1-ethyl-5-(naphthalen-1-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[5-(4-chloro-3-methyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
2-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyrimidine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-[2-(dimethylamino)ethyl]-8-(4-ethyl-5-methylpyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[2-(methylsulfanyl)phenyl]methyl}amine
6-methyl-2-(pyridin-3-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrimidin-4-amine
4-(2-methylphenoxy)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine-4-carboxylic acid
4-(4-{[4-(3-methylphenyl)phenyl]carbamoyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
(8R,9aS)-2-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
2-methyl-4-phenyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
N-[3-(3-fluorophenyl)phenyl]-1-(quinolin-2-ylmethyl)piperidine-4-carboxamide
2-(2,3-difluorophenoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
4-(azonan-1-yl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
4-(6-fluoro-1H-1,3-benzodiazol-2-yl)-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methoxyphenyl)methyl]acetamide
N-(oxolan-2-ylmethyl)-3-phenyl-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1,2-oxazole-5-carboxamide
1-methyl-1'-(2-propyl-1,3-thiazole-4-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropan-1-amine
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
1-benzyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]methyl}benzonitrile
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-N-(1,2-oxazol-3-ylmethyl)acetamide
(2S,4S)-4-amino-1-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-(2-{4-azaspiro[2.5]octan-4-ylmethyl}-6-methoxyphenoxy)propanoic acid
4-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-1-methyl-1,2,3,4-tetrahydroquinolin-2-one
2-(5-{4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
(1,4-dioxan-2-ylmethyl)(methyl)[(2-phenyl-1H-imidazol-4-yl)methyl]amine
2-ethyl-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(2,3-dihydro-1H-inden-2-yl)-8-[(3-hydroxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,4R)-1-({[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}methyl)-7,7-dimethylbicyclo[2.2.1]heptan-2-one