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N-[1-(dimethylamino)-2-methylpropan-2-yl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
1-methyl-4-[1-(propan-2-yl)piperidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-methoxy-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
ethyl 1-(2-hydroxyethyl)-5-{[4-(methoxycarbonyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
11-{[2-(2-fluorophenyl)ethyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
6-(3-methoxyphenyl)-N-[(3-methylpyridin-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 5-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-5-oxopentanoate
3-(5-methyl-1,2,4-oxadiazol-3-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
methyl 1-(2-methoxyethoxy)-2-oxo-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
N-benzyl-2-[4-(4-{[(3-chlorophenyl)methyl]amino}piperidin-1-yl)phenyl]acetamide
N-butyl-6-(2-chlorophenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
9-(4-methyl-1H-imidazole-2-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-2-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]azepane
3-[2-(dimethylamino)ethyl]-5-{1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1H-pyrazole-4-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]pyrrolidine-2-carboxamide
2-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)benzoic acid
(2S)-2-{[(3-cyano-4-methylphenyl)carbamoyl]amino}-3-methylbutanamide
[2-(dimethylamino)ethyl](methyl)(2-{[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]oxy}hex-5-en-1-yl)amine
10-methoxy-5-{[5-(oxan-2-yl)furan-2-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(3S,4S)-4-cyclopropyl-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(5-methoxy-1H-indol-2-yl)methyl]propanamide
{[2-(furan-2-yl)phenyl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
5-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrazin-2-ol
2-{5-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-4-phenyl-1H-imidazol-1-yl}acetamide
7-cyclohexyl-2-[(2,6-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[(4-methoxyphenyl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2-{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-2-yl}ethyl)morpholine
4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-[2-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}-6-ethoxyphenol
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-(pyridin-4-yl)piperazine
1-benzyl-N-methyl-5-[2-(pyridin-3-yl)acetyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-{4-[(3-cyanophenyl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
8-(1,3-dihydroxypropan-2-yl)-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 1-(2-methyl-1,3-thiazole-4-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-methoxyethyl 2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
1-methyl-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}urea
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
8-fluoro-2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]quinoline
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-methyl-1H-indole-6-carboxamide
2-(phenylamino)-N-[3-(phenylsulfanyl)propyl]pyrimidine-5-carboxamide
N-[(2-phenylphenyl)methyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-(2-acetylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-{[3-(cyclopentyloxy)phenyl]methyl}-3-(hydroxymethyl)pyrrolidin-3-ol
N4-[2-(1H-imidazol-4-yl)ethyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide