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4-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-1-methylpyrrolidin-2-one
3-[2-(4-chlorophenoxy)ethyl]-4-methoxy-N-methylbenzamide
6-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4-methylphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
4-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
7-[(5-methylfuran-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}[(3-fluorophenyl)methyl]amine
1-(4-methylpiperazin-1-yl)-3-(4-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)propan-2-ol
5-chloro-N-[(3-hydroxypyrrolidin-3-yl)methyl]-3-phenyl-1H-indole-2-carboxamide
3-(4-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
1-(cyclohex-3-ene-1-carbonyl)-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-(2,4-difluorophenoxy)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
methyl 8-benzyl-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(2-methyl-1,3-thiazole-5-carbonyl)-2-(2-phenylethyl)piperidine
3-(3-methoxyphenyl)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]ethan-1-one
N'-(5-methyl-1,2-oxazol-3-yl)-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]ethanediamide
2-[3-(propan-2-yl)-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazol-1-yl]pyridine
{3-[2-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]propyl}dimethylamine
3-[2-(4-chlorophenyl)morpholine-4-carbonyl]-2-methylphenol
4-methoxy-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-[(3-methylpyridin-2-yl)methyl]-4-[(3-methylthiophen-2-yl)methyl]piperazine
3-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}phenol
1'-(5-chloropyridine-3-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aR,7aS)-1-(2-methoxyacetyl)-4-(4-methoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2-(3-chlorophenyl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N5-[2-(3-fluorophenyl)ethyl]-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-N3-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
(3aR,6aR)-2-cyclobutanecarbonyl-5-(2,3-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
8-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 4-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-amido}piperidine-1-carboxylate
4-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-6-methyl-2-(pyridin-3-yl)pyrimidine
4-[(1-cyclohexylpropan-2-yl)amino]-N,N-dimethylbutanamide
N-[2-(pyridin-4-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,9aR)-8-(4-chlorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-(6-methoxypyrimidin-4-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(dimethylamino)ethyl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
N-(furan-2-ylmethyl)-2-{3-[3-(pyridin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
1-(furan-2-ylmethyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
5-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
(1R,5R)-6-benzyl-3-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
2-(4-fluorophenoxymethyl)-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1,3-oxazole-4-carboxamide
2-(cyclopropylmethyl)-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-(3,3-diphenylpropyl)-1-methylazepane-2-carboxamide
N-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-(1-methylpiperidin-4-yl)-6-oxo-N-(2-phenylethyl)-1,6-dihydropyrimidine-5-carboxamide