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{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
4-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-(ethoxymethyl)-1H-1,2,4-triazol-1-yl)-1-methylpiperidine
6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(3-chloro-4-propanamidophenyl)-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-(4-benzoylpiperazin-1-yl)-2-methyl-3-[methyl(propan-2-yl)amino]propan-1-one
N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-(trifluoromethyl)benzamide
3-chloro-4-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]phenol
2-{[3-(3-chlorophenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-ethylpyridine
5-{3-[(2-methoxyphenyl)methyl]-1-(4-methylphenyl)-1H-1,2,4-triazol-5-yl}piperidin-2-one
1-(adamantan-1-yl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazine
2-chloro-N-(1-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]benzamide
4-hydroxy-2-(3-methylphenyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidine-5-carboxamide
N-{[1-(diphenylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]pyridin-4-yl}methanol
4,4,4-trifluoro-1-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methoxyphenyl)ethyl]acetamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[3-(1H-imidazol-1-yl)propyl]pyrrolidin-2-one
2-(3,4-dimethoxyphenyl)-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
5-tert-butyl-3-[5-(cyclopentylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1H-pyrazole
1-{1'-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1,7,7-trimethyl-4-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]bicyclo[2.2.1]heptan-2-ol
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[3-(piperidine-1-carbonyl)phenyl]urea
4-methyl-5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,3-thiazol-2-amine
3-[5-(1-acetylpiperidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-(cyclopropylmethyl)-5-{imidazo[1,2-a]pyridine-2-carbonyl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(3-methoxyphenyl)sulfanyl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
5-methyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(methylamino)pyrimidine-5-carbonyl]pyrrolidine-3-carboxylic acid
2-methyl-4-[4-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)phenyl]butan-2-ol
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidine
2-{2-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(methoxymethyl)-1H-1,2,4-triazole
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
4-[(oxan-4-yl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
methyl 2-(4-{2-[(pyridin-3-ylmethyl)carbamoyl]ethyl}piperidine-1-carbonyl)benzoate
6-{3-oxo-3-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propyl}-2,3-dihydropyridazin-3-one
4-[1-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)ethyl]morpholine
9-[4-(1H-imidazol-1-yl)butanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-phenyl-4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine
7-methoxy-1-methyl-3-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
1-{2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-[2-(pyridin-2-yl)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
methyl 1-[(3S,5S)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[(3-methoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3-(4-fluorophenyl)-1H-pyrazole