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4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}thiomorpholine
N-[2-(dimethylamino)ethyl]-3-fluoro-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)benzamide
3-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
(4-{[1-(1H-indazole-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine
3,6-dimethyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1,2,3,4-tetrahydronaphthalene-2-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-methyl-3-phenyl-1H-pyrazole-5-carboxamide
1-methyl-N-[(1-phenylcyclohexyl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(pyrrolidin-1-ylmethyl)piperidine
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
8-{[4-(thiomorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
2-chloro-N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}pyridine-4-carboxamide
3-(1H-1,2,3,4-tetrazol-1-yl)-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
5-[2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carbonyl]-2-tert-butylpyrimidin-4-ol
2-{1-cyclopentyl-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
2-(1-{[1-(thian-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
2-(2-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-2-oxoethyl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)amine
3-chloro-4-[(1-cycloheptanecarbonylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
2-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
(3S,4S)-1-[(cyclohexylmethyl)carbamoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-[5-(1H-indole-6-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-[4-(benzyloxy)piperidine-1-carbonyl]-N,N-dimethylaniline
1-{2-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamido]ethyl}piperidine-3-carboxamide
1-{5-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
N,2-dimethyl-N-{[4-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
2-(3-methylbutyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
1-(cyclohexylmethyl)-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
1-[(3-methoxyphenyl)methyl]-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
2-methyl-5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
(3R,4S)-1-(3-chloro-4-propoxybenzoyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine
2-(3-chloro-2,4-difluorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
4-({2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
methyl (2S)-1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-2-carboxylate
5-fluoro-2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-4-amine
N-cyclopropyl-4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazine-2-carboxamide
3-[5-(cyclobutylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(morpholin-4-yl)propan-1-one
1'-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-methoxypropyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2-dihydroquinolin-2-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-cyclohexyl-3-hydroxy-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)propanamide
4-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}pyrimidin-2-amine