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(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
4-(cyclohexylmethyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-N,N-dimethylpyrrolidin-3-amine
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-amine
1-{3-oxo-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
methyl({[3-(4-methyl-1,4-diazepane-1-carbonyl)-1,2-oxazol-5-yl]methyl})(2-phenylethyl)amine
N-[3-(5-ethylpyrimidin-2-yl)phenyl]acetamide
4-{5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
3-(1H-1,3-benzodiazol-2-yl)-N-(1-ethyl-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
2-(2-fluoro-3-methylphenyl)-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[(E)-2-phenylethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-chloro-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-[(2-hydroxyethyl)(methyl)amino]-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
N-(1,2-oxazol-3-ylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
8-(2-methylpyridin-4-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopentyl-2-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-{2-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-[2-(diethylamino)-2-(furan-2-yl)ethyl]-1-[5-methyl-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(1,2,2-trimethylpyrrolidin-3-yl)methyl]acetamide
3-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methanesulfonyl-1,4-diazepane
N-benzyl-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-1,3-oxazole-4-carboxamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-ol
N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
2-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyridine-3-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-(2-amino-6-methoxypyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-benzyl-4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
2-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-(piperidin-4-yl)pyrimidin-4-amine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]acetamide
5-(morpholin-4-ylmethyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}furan-3-carboxamide
N-(2-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]morpholin-2-yl}ethyl)acetamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
(1R,9S)-5-amino-12-methyl-3-[4-(pyridin-2-yl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
(1R,2S,6R,7S)-4-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
1-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
N-[2-(5-methyl-4-{[3-(3-methyl-1H-pyrazol-1-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]benzamide
3-{[1-(propan-2-yl)piperidin-4-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(3,3-dimethylbutanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(2-methyl-1H-imidazol-1-yl)propanamide
N-{3-[4-(hydroxymethyl)phenyl]phenyl}cyclopropanecarboxamide
3-[(7-chloro-4-methylquinolin-2-yl)amino]-1-methylpyrrolidin-2-one
2-[4-(oxan-4-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazole
6-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
4-methyl-6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine