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4-{1-[2-methyl-2-(morpholin-4-yl)propanoyl]piperidin-3-yl}benzoic acid
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2S)-2-({2-[ethyl(phenyl)carbamoyl]ethyl}amino)-3-methylbutanamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(4-phenylbenzoyl)piperidin-1-yl]propan-1-one
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-chloropyridine-3-carboxamide
3,6-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-benzyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,3-thiazole-4-carboxamide
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methylpropanamide
2-(4-chloro-2-methylphenoxy)-N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]acetamide
ethyl 1-{3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperidine-3-carboxylate
6-methyl-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
(3R,4R)-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
(1-{[1-(4,5-dimethylthiophene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
1-[4-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
4-(2-fluoro-5-methylphenoxy)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-4-phenylpyridine
N-ethyl-3-methyl-4-[({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}carbamoyl)amino]benzamide
2-methyl-6-[4-(2-phenylethyl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(1,4-dioxan-2-ylmethyl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-1,3-oxazole-4-carboxamide
7-(3,3-diphenylpropanoyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-6-phenylpyridine-3-carboxylic acid
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-ol
4-{2-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-2-yl]ethyl}morpholine
(2E)-N-(3-hydroxy-3-methylbutyl)-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(3-methylbut-2-en-1-yl)piperazin-2-one
3-(2-benzyl-3-oxopiperazine-1-carbonyl)-4-fluorobenzene-1-sulfonamide
5-{5-methylthieno[2,3-d]pyrimidin-4-yl}isoquinoline
4-fluoro-3-{4-[2-(morpholin-4-yl)ethyl]piperazine-1-carbonyl}benzene-1-sulfonamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-chloropyridine
2-{4-[(2E)-3-phenylprop-2-en-1-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
1,3-dimethyl-2,6-dioxo-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl[2-(2-methyl-1H-indol-1-yl)ethyl]{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-benzyl-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
5-ethyl-2-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
{4-[(2-methoxynaphthalen-1-yl)methyl]-1,4-oxazepan-6-yl}methanol
4-methyl-6-{4-[4-(1,3-thiazol-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidin-2-amine
2-amino-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-cyclopropanecarbonyl-4-[4-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine
N'-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylbutanediamide
N-{[1-(isoquinolin-5-ylmethyl)piperidin-3-yl]methyl}cyclobutanecarboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methylacetamide
2-(2-methoxyethyl)-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}morpholine
5-(4-acetylphenoxymethyl)-N-methyl-N-[(1S)-1-phenylethyl]-1,2-oxazole-3-carboxamide
N-(2-methoxy-5-methylphenyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperazine
3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide