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5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]-4-{1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}pyrimidine
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2,5-dimethoxybenzamide
1-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-4-phenylpiperidin-4-ol
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-ol
1-ethyl-N-(3-methyl-1,2-thiazol-5-yl)-6-oxopiperidine-3-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-[(2-propylpyrimidin-5-yl)methyl]pyrrolidine-3-carboxylic acid
N-{4-[2-amino-3-cyano-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridin-4-yl]phenyl}acetamide
3-{4-[(6-chloropyridin-3-yl)methyl]piperazine-1-carbonyl}piperidine-1-carboxamide
3-(3-fluoro-5-methylphenyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazine
3-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-1-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]urea
2-({1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
5-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2,4,6-trimethyl-3-{[(2-methylbutan-2-yl)amino]methyl}phenyl)methanol
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-[(4-methoxypyridin-2-yl)methyl]urea
2-(2-methyl-1,3-thiazol-4-yl)-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}acetamide
4-(pyridin-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
3-[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)carbamoyl]pyridin-1-ium-1-olate
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzamide
3-amino-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]benzamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepane
5-(methoxymethyl)-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)furan-2-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
dimethyl(2-{4-[4-(propan-2-yloxy)benzoyl]morpholin-2-yl}ethyl)amine
1-(azepan-1-yl)-3-[3-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
3-(1,2,3,6-tetrahydropyridin-1-yl)-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
2-methyl-4-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-1,3-benzodiazole
4-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
1-(2-methanesulfonylethyl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazine
1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
8-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)piperidin-3-yl]benzoic acid
4-({3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-3-(4-chlorophenyl)-1H-pyrazole
N-[(4-phenyloxan-4-yl)methyl]pyrimidin-4-amine
2-[(3,5-difluorophenyl)methyl]-8-[(3E)-pent-3-enoyl]-2,8-diazaspiro[4.5]decan-3-one
4-{1H-pyrrolo[2,3-b]pyridin-4-yl}thieno[2,3-d]pyrimidine
1-ethyl-4-[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazole
2-(2-phenylethyl)-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
1-butyl-1-[(4-chlorophenyl)methyl]-3-(1,3-dimethyl-1H-pyrazol-4-yl)urea
8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclopropanecarbonyl-8-(4-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
1-(2-methoxyethyl)-8-(pyridin-2-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
2-hydroxy-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-4-(methylsulfanyl)butanamide
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-5-propyl-1,2-oxazole-4-carboxamide
4-(2-fluoro-3-methoxyphenyl)-2-methyl-1H-imidazole