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1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]piperidine-4-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-(1,3-benzothiazol-5-yl)-1-{[1-(morpholin-4-yl)cycloheptyl]methyl}urea
4-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(phenylformamido)acetamide
1-(1-benzothiophen-2-ylmethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
4-(propan-2-yl)-2-[4-(pyridin-4-yl)piperazin-1-yl]pyrimidine
[(1-cyclopentylpiperidin-4-yl)methyl]({[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-(2-ethoxyethyl)-5-(piperidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[(2,3-difluorophenyl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-(5-chloro-3-fluoropyridin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-benzyl-N-(oxan-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-({1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-N-[(6-methylpyridin-2-yl)methyl]benzamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
N-(furan-2-ylmethyl)-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
6-[4-(propan-2-yl)piperazin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(oxan-4-yl)piperazin-1-yl]ethan-1-one
(2S,4R)-4-amino-N-ethyl-1-{[4-(pyridin-2-yl)phenyl]methyl}pyrrolidine-2-carboxamide
1-(2-methoxyethyl)-4-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)pyrrolidin-2-one
(4aS,7aR)-1-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-2-(2-methylphenyl)-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
N-{2-[(4-fluorophenyl)formamido]ethyl}-3-(1-methylpiperidin-2-yl)propanamide
4-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-(oxolan-3-ylmethyl)-4-(1H-pyrrole-2-carbonyl)piperazine
(2R)-N1-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)pyrrolidine-1,2-dicarboxamide
1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperazine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
N-benzyl-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-sulfonamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-3-(trifluoromethyl)benzene-1-sulfonamide
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
(3S,9aR)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(4,6-dimethylpyridin-2-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
1-propyl-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
methyl 4-({3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)benzoate
(2R)-2-amino-3-(1H-indol-3-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
1-ethyl-4-[5-(2-fluorophenyl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(2-phenylethyl)amino]methyl}piperidin-2-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-indol-3-yl)propanamide
1-[(2S,4S)-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
2-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-cyclopentylpropanamide
N-[2-(dimethylamino)ethyl]-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
1-(2-methanesulfonylethyl)-5-methyl-5-phenylpiperidin-2-one
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(2,3,6-trifluorophenyl)ethan-1-one