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4-[1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]pyridine
3-methoxy-2-({4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(2-methylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
3-methyl-1-(4-methyl-2-oxo-2H-chromen-7-yl)-3-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-4-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(4-methoxy-2-methylphenyl)methyl]pyrrolidin-3-yl]methanol
4-(2-methoxyethyl)-1-(4-methylquinolin-2-yl)piperidine-4-carboxylic acid
3-{5-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}acetamide
N-(2,5-difluorophenyl)-2-{4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}acetamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-6-chloropyridazin-3-amine
N-cyclopropyl-4-methoxy-2-({1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
1-methyl-4-(1-methyl-4-phenylpiperidine-4-carbonyl)piperazine-2-carboxylic acid
N-[(5-methylpyrazin-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(4R)-3-methyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-1,3-thiazolidine-4-carboxamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
1-(2-fluorophenyl)-3-(2-methoxyethyl)-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
2-amino-6-(3,5-difluorophenyl)-4-(5-hydroxy-2-methoxyphenyl)pyridine-3-carbonitrile
2-(cyclohex-3-en-1-yl)-1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-imidazole
2-methoxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
5-(methoxymethyl)-N-[(2,3,6-trifluorophenyl)methyl]thiophene-2-carboxamide
2-{4-[(6-ethoxyquinolin-2-yl)methyl]piperazin-1-yl}-N-ethylacetamide
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
2-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}-3,5-dimethoxybenzoic acid
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-methanesulfonyl-N,4-dimethyl-N-[(2-methylphenyl)methyl]quinazolin-2-amine
2-[({[2-(benzylamino)pyrimidin-5-yl]methyl}(methyl)amino)methyl]-3,4-dihydroquinazolin-4-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-cyclopentylpiperazin-2-one
4-[4-(4-cyclopropanecarbonylpiperazin-1-yl)-6-methylpyrimidin-2-yl]morpholine
(3S,4S)-3-{[1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-4-hydroxy-1λ6-thiolane-1,1-dione
N-(3,4-dimethoxyphenyl)-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
N-({4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-4-(trifluoromethyl)benzamide
1-methyl-N-[(1-methyl-1H-indol-5-yl)methyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
2-methyl-2-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)propanamide
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
3-(4-methyl-1,3-thiazol-5-yl)-1-[(2S)-2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]propan-1-one
3-methoxy-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(4-fluoro-2-methylphenyl)ethan-1-one
4-(1H-indole-6-carbonyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
4-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-[(1S,5R)-6-[(3-hydroxy-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
5-[(1-benzothiophen-5-ylformamido)methyl]-N-methylfuran-2-carboxamide
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(4aS,8aR)-2-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-decahydroisoquinoline
1-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
7-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-methoxyphenyl)-3-methyl-5-[2-(methylsulfanyl)ethyl]-1H,4H-pyrazolo[3,4-d]imidazole
3-(4-chlorophenyl)-5-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole