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2-[(3,5-difluorophenyl)methyl]-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
(2S)-1-[(1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidine-2-carboxamide
2-ethyl-4-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
2-(3-chloro-4,5-diethoxyphenyl)-1-(pyrrolidin-3-yl)-1H-imidazole
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclopropanecarboxamide
7-methyl-4-[2-(2-methyl-1,4-oxazepan-4-yl)-2-oxoethyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-(thiophen-3-yl)acetamide
5-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-(3,3-diphenylpiperidine-1-carbonyl)pyridine-2-carbonitrile
4-chloro-2-{[methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-methanesulfonamidopropanamide
3-[(2R,3R,6R)-5-(1H-indazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2E)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-phenylprop-2-enamide
2-{3-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
1-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]pyrimidin-2-amine
4-[5-(dimethyl-1,2-oxazol-4-yl)thiophen-2-yl]-1,3-thiazol-2-amine
[4-(5-propyl-1,2-oxazole-3-carbonyl)morpholin-3-yl]methanol
6-(dimethylamino)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)pyridine-3-carboxamide
2-{2-[(2-ethylmorpholin-4-yl)methyl]-4-(pyridin-3-yl)phenoxy}acetic acid
1-[(3-methoxyphenyl)methyl]-4-(3-methylthiophene-2-carbonyl)piperazin-2-one
1-[1-(6-ethylpyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxan-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(quinolin-4-ylmethyl)-1,4-diazepan-6-yl]oxy}acetamide
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-[(dimethylcarbamoyl)amino]acetamide
(2S,4R)-4-(dimethylamino)-1-(2,6-dimethylquinoline-4-carbonyl)pyrrolidine-2-carboxylic acid
6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-7-methyl-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-hydroxy-2-(4-methylphenyl)-N-{3-[(pyridin-3-yl)amino]propyl}pyrimidine-5-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)morpholine-4-carboxamide
1-[(2-chloro-5-fluorophenyl)methyl]-4-(1-methylpiperidin-4-yl)piperazine
methyl 4-[(3-{2-[(3,5-dimethoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
1-[(5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-2-methoxyphenyl)methyl]pyrrolidine
ethyl 4-({1-[(4-methoxyphenyl)methyl]-7-oxoazepan-4-yl}amino)piperidine-1-carboxylate
4-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]phenol
N-cyclopentyl-6-[3-(morpholin-4-ylmethyl)phenyl]pyridazin-3-amine
5-amino-3-[4-hydroxy-3-(prop-2-en-1-yl)phenyl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
(3S,4S)-4-cyclopropyl-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(oxan-4-yl)benzamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-methylpyrimidine
5-benzyl-4-(2-methoxyethyl)-1-(4-methylphenyl)piperazin-2-one
2-{[4-(3-chlorophenyl)-5-[(propan-2-yloxy)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-amine
1-methyl-2-oxo-8-[(4-phenylphenyl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-[(2-methyl-1H-imidazol-4-yl)methyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(azepan-1-yl)-N-[3-(1H-1,3-benzodiazol-2-yl)propyl]acetamide