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N-(2-acetamidophenyl)-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(1,1-dioxo-1λ6-thiolan-3-yl)piperidine-4-carboxamide
2-[5-(1-benzothiophen-3-yl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-methyl-1,3-benzothiazole-5-carboxamide
2-{4-cyclobutyl-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-carbamoylcyclopentyl)-4-(4-chlorophenoxy)piperidine-4-carboxamide
(2,1,3-benzothiadiazol-4-ylmethyl)(benzyl)(1,3-thiazol-2-ylmethyl)amine
2-methyl-4-[4-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)phenyl]butan-2-ol
2-cyclopentyl-8-(5-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(2-ethyl-1H-imidazol-1-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
N5-cyclopropyl-N6-(thiophen-2-ylmethyl)-N5-[(trimethyl-1H-pyrazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4,6,7-trimethyl-2-{4-[(2,4,5-trimethoxyphenyl)methyl]-1,4-diazepan-1-yl}quinazoline
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-{4-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
5-chloro-2-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}phenol
5-butyl-1'-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(dimethylamino)ethyl]amine
1-[(2-fluorophenyl)methyl]-4-(piperidin-4-ylmethyl)-1,4-diazepane
3-[4-(3-methylphenyl)piperazin-1-yl]-1-(1,4-oxazepan-4-yl)propan-1-one
2-acetamido-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
N-benzyl-6-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)benzoic acid
methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
4-(2,6-dimethylpyridin-3-yl)-N-[3-(1H-imidazol-1-yl)butyl]pyrimidin-2-amine
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(methylsulfanyl)ethan-1-one
1-[2-(trimethyl-1H-pyrazol-1-yl)acetamido]cyclopentane-1-carboxamide
(3S,4S)-4-cyclopropyl-1-(1-phenylpiperidin-4-yl)pyrrolidine-3-carboxylic acid
N-[(1S,2R)-2-aminocyclobutyl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
5-{1-[2-methyl-5-(trifluoromethyl)benzoyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
3-({2-[1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
(3S,4S)-4-methyl-1-[1-(4-methylbenzenesulfonyl)azetidin-3-yl]piperidine-3,4-diol
5-methyl-1'-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}benzoic acid
2-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
4-cyano-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]oxane-4-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylacetamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-methyl-N4-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
1-(5-methyl-1,3,4-oxadiazol-2-yl)-3-(thiophene-2-carbonyl)piperidine
(2S)-N-{3-[(3-methoxyphenyl)carbamoyl]phenyl}-5-oxopyrrolidine-2-carboxamide
N-[(3-ethoxyphenyl)methyl]-4-methanesulfonyl-N-(prop-2-en-1-yl)benzamide
methyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(trifluoromethyl)phenyl]methyl}amine
5-ethyl-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-pyrazole
2-{[(3-cyano-6-methylpyridin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
[(2S,4R)-1-[(5-chlorofuran-2-yl)methyl]-4-(dimethylamino)pyrrolidin-2-yl]methanol