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[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-[(3-ethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)cyclopropanamine
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-(1-methyl-1H-pyrazol-5-yl)-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
N-[(3-methoxyphenyl)methyl]-N-methyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1'-[(3-chloro-2-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-[5-(1-ethylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methylpropan-1-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[(3-ethoxy-3-oxopropyl)carbamoyl]piperidine-3-carboxylate
2-{4-[3-(1H-pyrazol-1-yl)propyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
methyl 5-(diethylsulfamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-[5-(1,4-dioxan-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N3-tert-butyl-N5-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-cyclopentyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N2-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N4-methylpyrimidine-2,4-diamine
(2S,4S)-4-(benzylamino)-1-[(3-chlorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
2-(4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
5-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
1-(4-chlorophenyl)-N-{[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
N-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridine-6-carbonyl]-1λ6-thiane-1,1-dione
2-(2-methylfuran-3-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-N,8-dimethyl-2-(1-phenyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-8-(4-methylpiperazine-1-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-(2H-1,3-benzodioxol-5-yl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetic acid
2-(5-acetylthiophen-3-yl)-N-[(2-fluorophenyl)methyl]acetamide
(2S,4S)-4-amino-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-3-carboxamide
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
1-(2,1,3-benzothiadiazol-4-yl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
N,N,4-trimethyl-3-({[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidin-2-one
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)furan-3-carboxamide
5-(3,4-difluorophenoxymethyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
(2S)-1-(4-acetyl-4-phenylpiperidin-1-yl)-2-amino-4-(methylsulfanyl)butan-1-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
N-{2-[(2-chlorophenyl)formamido]ethyl}-3-(pyridin-4-yl)propanamide
N-[3-(4-acetyl-4-phenylpiperidin-1-yl)-3-oxopropyl]methanesulfonamide
1-[(2-chlorophenyl)methyl]-3-phenylpyrrolidin-3-ol
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[3-(3-fluorophenyl)phenyl]piperidin-4-amine
1-{1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-3-methylbutan-1-ol
1-(dimethyl-1,3-thiazol-2-yl)-3-(oxan-4-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
ethyl 4-(2-phenylethyl)-1-(quinoxalin-5-ylmethyl)piperidine-4-carboxylate
methyl (2S,4R)-1-{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}-4-(dimethylamino)pyrrolidine-2-carboxylate
6-(1-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one