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N,3-dimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1,2-oxazole-5-carboxamide
7-cyclobutaneamido-N-[(2-fluorophenyl)methyl]-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
2-[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
3-benzyl-4-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperazin-2-one
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-3-(trimethyl-1H-pyrazol-1-yl)propanamide
4-[2-(2-methoxyphenyl)acetyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2,3-dimethyl-7-(4-methylpyrimidine-5-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(2-chloro-4-fluorophenoxymethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-(3-methoxybenzoyl)piperazine
6-(methoxymethyl)-2-(3-{[3-oxo-2-(propan-2-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-({[(2,5-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
methyl(piperidin-4-ylmethyl)[1-(pyridin-4-yl)ethyl]amine
5-{2-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
6-(4-ethylphenyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(3,5-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S)-1-{2-[4-(4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-(1-propylpiperidin-4-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}acetamide
2-fluoro-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5-sulfamoylbenzamide
1-[1-(2-fluorobenzoyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(3,5-difluorophenyl)ethyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-phenyl-N-[(3R)-pyrrolidin-3-yl]adamantane-1-carboxamide
4-(4-fluorophenyl)-4-oxo-N-(oxolan-3-yl)butanamide
(3S,4R)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-4-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
5-(3-methylbut-2-en-1-yl)-1'-(pyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-{[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-[2-(dimethylamino)-2-(4-fluorophenyl)-N-methylacetamido]-N-methylpropanamide
2-[(ethylamino)methyl]-4-(6-methoxypyridin-2-yl)phenol
1'-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
N-[1-(pyrazin-2-yl)propan-2-yl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
4-ethyl-4-({[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]amino}methyl)hexanenitrile
N-methyl-N-(oxan-2-ylmethyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(furan-3-ylmethyl)propanamide
1-(oxan-4-ylmethyl)-4-[2-(pyridin-2-ylsulfanyl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
3-(3-fluorophenyl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazole-4-carboxamide
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-4-(1H-pyrrol-1-yl)phenol
N-(2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)-4-ethylcyclohexane-1-carboxamide
methyl[3-(1H-pyrazol-1-yl)propyl](quinolin-4-ylmethyl)amine
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-3H,4H-pyrido[2,3-d]pyrimidin-4-one
8-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(3R,4R)-1-{[3-(2-aminoethyl)phenyl]methyl}-4-(azepan-1-ylmethyl)pyrrolidin-3-yl]methanol
4-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-N,N-dimethylaniline
1-[(3-chlorophenyl)methyl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide