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N-[(2S)-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl]acetamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-[(3E)-pent-3-enoyl]pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[4-(1-methyl-1H-indole-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
(1R,5S)-6-(4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)-6-azabicyclo[3.2.1]octane
N,8-dimethyl-2-propyl-N-(pyrimidin-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(pyrimidin-4-ylmethyl)acetamide
1-{1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}cyclopropane-1-carboxamide
1-[(2R)-oxolane-2-carbonyl]-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-ethyl-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxylic acid
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
[4-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)quinazolin-2-yl]methanol
N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(4-chlorophenyl)-N-cyclopropyl-3-phenylpropanamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-methoxyquinoline-4-carboxamide
3-(2-methoxyphenyl)-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}propanamide
[(3R,4S)-1-{[4-(methylsulfanyl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-{4-[3-(2-fluorophenyl)pyrrolidin-1-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
1-[4-(3-fluorophenyl)phenyl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidin-4-amine
3-(3-methoxypropyl)-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(methylamino)pyrimidine-5-carboxamide
1-(1H-imidazol-4-ylmethyl)-2-(3-methoxyphenyl)piperidine
5-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-(ethoxymethyl)-1-ethyl-1H-1,2,4-triazole
3-cyclopropyl-1-[(4-fluorophenyl)methyl]-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazole
2-[2-methyl-3-({[1-(1H-pyrazol-1-yl)propan-2-yl]amino}methyl)-1H-indol-1-yl]acetamide
ethyl 1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
(3S,4R)-4-(3-fluorophenyl)-1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
5-(3-methylpyridin-2-yl)-2-(thiophen-2-yl)-1,3-benzoxazole
N-methyl-2-(methylamino)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(2-hydroxyethyl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
2-[9-(2,3-difluorobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-[1-(4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]propan-1-one
N-[2-(4-chlorophenyl)propyl]-3-[(2-fluorophenyl)formamido]propanamide
2-(furan-2-yl)-N-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]azepane-1-carboxamide
(2S,4S)-4-amino-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
2-oxo-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(propan-2-yl)acetamide
2-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(4-methoxy-3-methylphenyl)-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-{1-[3-(methylsulfanyl)propyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperazine-1-sulfonamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
(4aR,7aS)-1-benzyl-4-(5-methylpyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 1-[(3R,5S)-1-[(4-hydroxyphenyl)methyl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1H-1,2,4-triazole-5-carboxamide