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2-(4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
N-methyl-2-[2-(morpholin-4-ylmethyl)phenyl]pyrimidin-4-amine
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-(2-phenylethyl)piperidine
3-(3-fluorophenoxymethyl)-5-(5-methoxyfuran-2-yl)-1-methyl-1H-1,2,4-triazole
5-methoxy-9-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
N-[1-(3-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
9-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(cyclohexylsulfanyl)propyl]-3-[3-(methylsulfamoyl)phenyl]urea
2-tert-butyl-6-(3-chloro-2-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
1-[1-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-4-yl)ethyl]-4-methylpiperazine
N-tert-butyl-2-[6-(pyrrolidin-1-yl)pyridazin-3-yl]benzene-1-sulfonamide
N-methyl-4-(4-methylphenoxy)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-4-carboxamide
2-(1H-1,2,3-benzotriazol-1-yl)-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
5-(3,4-difluorophenoxymethyl)-3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,2-oxazole
7,7-dimethyl-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}pyrimidin-4-yl)piperidin-4-ol
6-[(diethylamino)methyl]-N-methyl-N-(1-methylpyrrolidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-ethyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}propanamide
1-(2-methoxyethyl)-4-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperazine
1-{4-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]piperazin-1-yl}ethan-1-one
3-(azocan-1-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}propanamide
2-cyclopropanecarbonyl-8-(1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclohexyl-2-(pyridin-3-yl)-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
(3aR,5R,6S,7aS)-2-[3-(3-hydroxy-3-methylbutyl)benzoyl]-octahydro-1H-isoindole-5,6-diol
1'-(oxolane-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-[(dimethylamino)methyl]piperidin-3-ol
3-[2-(4-fluorophenyl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
8-(2,1,3-benzoxadiazol-4-ylmethyl)-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-[3-oxo-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperazin-2-yl]acetate
7-(2,3-dichlorobenzenesulfonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-(3-oxopiperazin-1-yl)acetamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
7-chloro-3-({[(2-fluorophenyl)methyl]amino}methyl)-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
(4aR,7aS)-1-benzyl-4-(2-ethoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrazine-2-carboxamide
1-[3-(methylsulfanyl)propyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
2-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazole
5-[(5-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}furan-2-yl)sulfanyl]-1H-1,2,4-triazole
2-[(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-2H-1,2,3,4-tetrazole
(4aR,7aS)-1-(2-methoxyacetyl)-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
1-[6-methyl-3-(1,4-oxazepan-4-ylmethyl)quinolin-2-yl]piperidin-3-ol
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}but-3-en-1-one
N2-[1-(3-phenylpropyl)piperidin-3-yl]pyrimidine-2,4-diamine
1-({5-[(4-chloro-2-fluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-({2-[(dimethylamino)methyl]phenyl}methyl)-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine