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ethyl 4-[(2-chlorophenyl)methyl]-1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[(E)-2-(2-methoxyphenyl)ethenyl]-1H-1,3-benzodiazole-6-carboxylic acid
4-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}benzoic acid
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[2-(cyclopent-2-en-1-yl)acetyl]piperidine-4-carboxylic acid
1-(2-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
5-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-2-ol
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[2-(morpholin-4-yl)ethyl]piperidin-4-amine
2-(2-{[cycloheptyl(methyl)amino]methyl}phenyl)-6-cyclopropyl-3,4-dihydropyrimidin-4-one
4-acetamido-2-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}benzamide
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
4-(4-fluorophenoxy)-1-(oxolane-3-carbonyl)piperidine
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2,3-dihydro-1H-imidazol-2-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(1,2-oxazinan-2-yl)pyridine-3-carboxamide
N4,N4,5-trimethyl-N2-[3-(oxolan-3-yl)propyl]pyrimidine-2,4-diamine
N-{[3-(difluoromethoxy)phenyl]methyl}-4-methylpyrimidine-5-carboxamide
4-ethenyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
2-[(2R)-2-hydroxypropanoyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-phenylpropan-1-one
2-methyl-4-{3-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}but-3-yn-2-ol
8-(1H-indol-3-ylmethyl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-ethyl-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(benzenesulfonyl)-4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazine
8-(2,4-dimethylpyrimidine-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N4-{[3-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
methyl 3-(oxolane-3-amido)-1-(2-phenylethyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-methyl-6-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
5-amino-3-(1-methyl-1H-imidazol-5-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-imidazole-4-sulfonamide
(2S)-2-{[6-(aminomethyl)pyrimidin-4-yl]amino}-3-cyclohexylpropan-1-ol
8-(oxane-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(methylsulfanyl)-6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-1H-1,3-benzodiazole
ethyl 1-(2-fluorophenyl)-5-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-1H-pyrazole-4-carboxylate
7-fluoro-3-methyl-2-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]-1H-indole
[1-(5-chloropyridin-2-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
2-[4-(1H-indol-2-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
(4aR,7aS)-1-(pyridin-4-ylmethyl)-4-[2-(pyrrolidin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(cyclopentylmethyl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1-methyl-1H-indazol-3-yl)-2-[4-(pyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
N-methyl-5-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)furan-2-carboxamide
[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-(2-methylpropyl)benzamide
3-methyl-8-{3-[methyl(1-methylpyrrolidin-3-yl)amino]propanoyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methanesulfonyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]benzamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-cyclopropyl-5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
N,N-dimethyl-2-[(1S,5R)-6-[(5-methylthiophen-2-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(2-methoxyphenyl)acetic acid
1-(2-ethoxyphenyl)-4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine