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2-methyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-dihydroquinolin-4-one
2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-4-(pyridin-2-yl)pyrimidine
4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]-1-(oxan-4-yl)piperidine
(2S,4S)-4-amino-N-methyl-1-{4-[(pyridin-4-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
N,4-dimethyl-4-[(4-propylpyrimidin-5-yl)formamido]pentanamide
1-{4-[6-hydroxy-4-(thiophen-3-ylmethyl)-1,4-diazepan-1-yl]piperidin-1-yl}ethan-1-one
(2S,4R)-4-(dimethylamino)-1-(2-phenylbenzoyl)pyrrolidine-2-carboxylic acid
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-(1H-indol-3-yl)ethyl]pyridin-2-amine
[2,2-dimethyl-3-(morpholin-4-yl)propyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
ethyl 5-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4-(trifluoromethyl)pyrimidin-2-amine
2-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)methyl]benzoic acid
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
2-(4-chlorophenyl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
2,3-dimethyl-6-[3-(propoxymethyl)pyrrolidine-1-carbonyl]quinoxaline
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-5-cyclopropyl-1,3-oxazole
methyl 2-[3-({3-[(furan-2-ylformamido)methyl]piperidin-1-yl}methyl)-1H-indol-1-yl]acetate
5-(2-chlorophenyl)-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]furan-2-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,3-oxazole-5-carboxamide
4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2-methylphenol
N-[5-chloro-2-(2-methylpiperidin-1-yl)phenyl]pyridazine-4-carboxamide
7-acetamido-2-(2-methoxyphenyl)-1-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(2S)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-acetamidopropanamide
2-(4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
N-(1H-imidazol-2-ylmethyl)-N,1,3-trimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}piperazine
ethyl 4-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}piperidine-1-carboxylate
2-(5-methyl-1H-pyrazol-1-yl)-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-[1-(3-methylbenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
5-(1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
2-(2-methylpropyl)-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(3-fluorophenyl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
4-[1-(3-methyl-1-benzothiophene-2-carbonyl)piperazine-2-carbonyl]morpholine
2-[2-(pyridin-2-yl)ethyl]-9-(trimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-methylpiperidin-2-yl)-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}propanamide
N-methyl-4-(4-methyl-2-phenylpiperazine-1-carbonyl)pyridin-2-amine
2-({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetic acid
6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N'-(2-methylphenyl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)propanediamide
2-{4-[(4-cyclopropanecarbonylpiperazin-1-yl)methyl]phenyl}-5,6-dimethyl-3,4-dihydropyrimidin-4-one
4-methoxy-2-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
4-[7-(2,6-dimethylbenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
(1R,5S,6S)-N-cyclopropyl-3-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-(4-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-methoxyphenol
N-[2-(morpholin-4-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(2S,4R)-4-amino-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
dimethyl({4-methyl-5-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one