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methyl 3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
N,N-dimethyl-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}azepan-4-amine
N-[(3-methylphenyl)methyl]-5-(piperazine-1-carbonyl)-1-propyl-1H-1,3-benzodiazol-2-amine
3-[2-(4-fluorophenyl)morpholin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole
N-(6-methylpyridin-3-yl)-1-(2-propylpyridine-4-carbonyl)piperazine-2-carboxamide
1-[5-(2-methylpyridine-3-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
N-[(4-acetylmorpholin-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
2-cyclohexyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-amino-4-ethyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,3-thiazole-5-carboxamide
2-{4-[(3-fluorophenyl)methyl]-3-oxopiperazine-1-carbonyl}-3,4-dihydroquinazolin-4-one
ethyl 1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
(2R,3R,6R)-5-[(5-methylfuran-2-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(3-methoxyphenyl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
3-{1-[(3,5-dimethoxyphenyl)methyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
N-[(2-methoxynaphthalen-1-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-cyclohexyl-5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopropyl-5-(2-ethoxypyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(4-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
(3S,4S)-4-cyclopropyl-1-(quinoxalin-2-yl)pyrrolidine-3-carboxylic acid
1-methyl-2-[5-(5-methyl-1,2-oxazol-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
7-chloro-4-(5-fluoro-2-methylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-propyl-N-(4H-1,2,4-triazol-4-yl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
1-ethyl-4-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methanol
2-benzyl-9-[4-(pyrrolidin-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-2-{[(3-phenoxypropyl)amino]methyl}quinolin-4-ol
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
2-(3-chloro-4-fluorophenoxy)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
1-(4-{4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3S,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperidin-4-ol
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2,3-dimethyl-1H-indole
ethyl({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(pyridin-4-ylmethyl)amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-methylpiperidine
3-(1,2-oxazinan-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]propanamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}propanamide
5-(propan-2-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
6-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-(2-phenoxyethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-(3-chloro-4-hydroxybenzoyl)-3-(hydroxymethyl)piperidin-3-ol
6-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
4-(4-chlorophenyl)-1-{[5-(2,5-dimethoxyphenyl)-2-hydroxyphenyl]methyl}piperidin-4-ol