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1-(2-benzylphenyl)-3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-methylurea
1-[(5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-methylpiperazine
1-[(2-fluorophenyl)methyl]-4-(pyridin-3-ylmethyl)piperazin-2-one
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one
7-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-ethyl-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(1R,3S,3aS,6aR)-5-ethyl-1-(1H-indol-3-ylmethyl)-3-(1-methyl-1H-imidazol-5-yl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
4-methyl-2-(propan-2-yl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,3-thiazole-5-carboxamide
5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
6-cyclopropyl-2-[4-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-{4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-6-methylpyrimidin-2-yl}phenol
1-[(2-methoxyphenyl)methyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
(4aR,7aS)-1-ethyl-4-[4-(trifluoromethyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)-3-methoxyphenol
1-(oxan-4-ylmethyl)-2-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazole
(5S,9aS,9bS)-5-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
1-(5-chloropyridin-2-yl)-4-(1-methylcyclopropanecarbonyl)-1,4-diazepan-6-ol
1-[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
2-{1-[1-(2,6-dimethylquinoline-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
1-[9-(cyclohexylmethyl)-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(1H-imidazol-4-yl)ethan-1-one
4-(2-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}ethyl)morpholine
5-methyl-1-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1-methanesulfonylpiperidin-4-yl)-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
2-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]benzonitrile
(4aS,7aR)-1-[(3-methylthiophen-2-yl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-tert-butyl-N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-(trifluoromethyl)pyrimidin-4-amine
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxylic acid
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}amine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-(2-hydroxyethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 5-{[(1R,3R)-3-aminocyclopentyl]carbamoyl}-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxylate
5-(furan-3-yl)-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-4-(4-methylphenyl)pyrimidin-2-amine
1-[4-(3-methylpyridin-4-yl)piperazin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
5-methyl-N-[1-(thiophen-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[1-(5-propylthiophene-3-carbonyl)azetidin-3-yl]pyridine
8-methoxy-2-{[1-(morpholin-4-yl)hex-5-en-2-yl]oxy}quinoline
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
6-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-3-phenylpyrazolo[1,5-a]pyrimidine
(3S,4R)-1-(8-fluoroquinoline-2-carbonyl)-4-methylpiperidine-3,4-diol
4-(2-chlorophenyl)-3-[2-(phenylamino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclohexyl-2-(dimethylamino)-2-(2-fluorophenyl)-N-(2-hydroxyethyl)acetamide
8-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{3-[3-(2-fluoro-4-methylphenyl)phenyl]-1H-pyrazol-1-yl}acetamide
5-methoxy-2-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]phenol
4-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-2-methylphenol
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-[2-(3-chlorophenyl)ethyl]-4-[(pyridin-3-ylmethyl)amino]pyrrolidin-2-one