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1-(5-methoxy-2-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
1-(cyclohexylmethyl)-N5-[(2-methoxyphenyl)methyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
N-ethyl-5-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidin-2-amine
2-{[(2-hydroxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amino]methyl}-5,8-dimethylquinolin-4-ol
(3S,4S)-4-(morpholin-4-yl)-1-{[2-(2-phenylethynyl)phenyl]methyl}pyrrolidin-3-ol
(2,1,3-benzoxadiazol-5-ylmethyl)({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
3-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)-1-(3-methoxypiperidin-1-yl)propan-1-one
2-(4-chlorophenyl)-4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethan-1-one
2-{[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
3-[(2R,3R,6R)-5-(2-ethylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
8-fluoro-2-({[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amino}methyl)quinolin-4-ol
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1,2-oxazole-3-carboxamide
N-cyclopentyl-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(4-{[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
4-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1-(3-methoxyphenyl)piperazin-2-one
7-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-1,4-oxazepane
1-({1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(propan-2-yl)pyridin-2-amine
4-[3-ethoxy-4-methoxy-5-(prop-2-en-1-yl)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2,5-dimethylfuran-3-carbonyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
3-(cyclopropylmethyl)-1-{2-[4-(dimethylamino)phenyl]acetyl}piperidine-3-carboxylic acid
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(thiophen-3-ylmethyl)piperidin-3-yl]propanamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-ol
N-(2-methoxyethyl)-4-methyl-3-[(phenylcarbamoyl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)cyclopropane-1-carboxamide
N2-cyclopropyl-N4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-butyl-8-(5-propyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-methyl-8-[2-(morpholin-4-yl)-2-oxoethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,3-benzothiazole-5-carboxamide
1-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-(furan-2-yl)ethane-1,2-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
N-(1-benzylpyrrolidin-3-yl)-2-cyclobutyl-5-(2-methoxyacetamido)-1-methyl-1H-1,3-benzodiazole-7-carboxamide
3-(azepane-1-carbonyl)-N-butyl-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-[2-(morpholin-4-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-({cyclohexyl[(4-fluorophenyl)methyl]carbamoyl}amino)phenyl]acetamide
(3aR,6aR)-2-(2-methoxyethyl)-5-[2-(methylsulfanyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-3-{[3-(methylsulfanyl)phenyl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-benzylpyrrolidin-3-yl)-3-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]propanamide
(4S)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazine
N-[3-({[1-(4-fluorophenyl)propan-2-yl]amino}methyl)-5-(4-methylpiperazine-1-carbonyl)phenyl]acetamide