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2-{2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2-oxoethyl}-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
4-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidine-1-carbonyl]oxane-4-carbonitrile
(2S,4S)-4-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-methylpyrrolidine-2-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
(3S)-3-ethyl-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]morpholine
[(1-ethyl-1H-pyrazol-4-yl)methyl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
N-{3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methoxy]phenyl}-4,6-dimethylpyrimidin-2-amine
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-benzyl-7-methoxy-N-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine-3-sulfonamide
5-(propan-2-yl)-3-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
8-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoline
6-(5-methyl-1H-indol-3-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-{[1-(2,3-dihydro-1H-inden-5-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}morpholine
(4S)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-3,3,4-trimethylpiperidin-4-ol
3-benzyl-8-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-hydroxy-N-[1-(4-methylpyridin-2-yl)propyl]-2-phenylpyrimidine-5-carboxamide
4-{1-[6-(piperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methyl-7-(methylsulfanyl)quinoline
3-fluoro-4-methoxy-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
1-tert-butyl-N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
5-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
N-(3-chloro-4-fluorophenyl)-3-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]propanamide
2-(pyridin-4-yl)-N-[1-(thiophen-2-yl)propan-2-yl]pyrimidine-5-carboxamide
5-(furan-3-yl)-3-(oxolan-3-yl)-1-phenyl-1H-1,2,4-triazole
1-(6-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridin-2-yl)ethan-1-ol
(3S,4S)-1-[(3-methylquinoxalin-2-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
1-{3-[(4,6-dimethylpyrimidin-2-yl)amino]piperidin-1-yl}-2-methylpropan-1-one
N-(furan-2-ylmethyl)-4-{[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amino}pyridine-2-carboxamide
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-2-(1H-pyrazol-1-yl)butanamide
[(1R,3S,3aS,6aR)-5-benzyl-3-(5-fluoro-2-methoxyphenyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-(3-chlorophenyl)-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}pyrrolidin-2-one
(4aS,7aR)-1-(3-hydroxy-4-methylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethyl-1,2-oxazol-4-yl)-1-(4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
5-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)-N-methylfuran-2-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-(quinoxalin-2-ylmethyl)-1H-pyrazole-4-carboxamide
4-[2-(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]morpholine
3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-{2-[2-(propan-2-yloxy)phenyl]ethyl}urea
9-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-ethyl-N-[(4-fluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidin-3-yl)piperazine
3-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
2-[(2R)-2-aminopropanoyl]-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-(3-methyl-1,2-oxazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{3-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1,3,4-thiadiazol-2-amine
4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-7-hydroxy-1,2,3,4-tetrahydroquinolin-2-one
6-methyl-5-(2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(1-butyl-1H-imidazol-2-yl)-1-(ethanesulfonyl)piperidine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methanol
5-(methoxymethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-2-carboxamide