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3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidin-3-yl]propan-1-ol
N-(1,3-dihydroxypropan-2-yl)-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-(hydroxymethyl)-1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-ol
2-amino-3-ethyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
7-{[5-(2-chlorophenyl)furan-2-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
6-ethyl-2-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-dihydropyridine-4-carboxamide
3-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}phenol
(1R,2R,4R)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
propan-2-yl 2-chloro-5-(6-oxopiperidine-3-amido)benzoate
3-(4-fluorophenyl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
6-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(thian-4-yl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-amino-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
N-[3-(3-methylphenyl)phenyl]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
3-[(dimethylamino)methyl]-N-(2-methoxy-6-methylphenyl)benzamide
N-cyclobutyl-3-{[(5-ethylpyridin-2-yl)methyl]sulfamoyl}benzamide
5-methoxy-1-methyl-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1H-indole-2-carboxamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]benzamide
(1S,5R)-3-benzyl-6-(propane-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(thiophene-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl (2S)-2-[(6-methoxypyrimidin-4-yl)amino]-2-phenylacetate
2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})amine
(3S)-1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-ol
(1S,6R)-9-[2-(trifluoromethoxy)benzenesulfonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
3-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-1-[5-(2-chlorophenyl)furan-2-carbonyl]-2-(methoxymethyl)pyrrolidine
4-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyridine
(1S,5R)-6-(2-methoxyethyl)-3-[(2E)-3-phenylprop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonane
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
1-(4-{[3-({1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)-4-methoxyphenyl]methyl}piperazin-1-yl)ethan-1-one
3-{1-[1-(2-hydroxyphenyl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenol
3-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-N-(oxolan-3-ylmethyl)benzamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
2,2,6,6-tetramethyl-4-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]piperidine
3,6-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(2-{1-[4-(methylsulfanyl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
ethyl 4-[2-(1-benzyl-3-oxopiperazin-2-yl)acetamido]piperidine-1-carboxylate
5-(2,2-diphenylacetyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[3-(dimethylamino)propyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N-ethyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-[4-(2-fluorophenoxy)phenyl]-1-(3-phenylprop-2-ynoyl)piperidine-4-carboxamide
3-ethyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1H-pyrazole-5-carboxamide
1-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3-benzotriazole
5-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-(piperidin-1-yl)propan-1-one