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9-[2-(1H-imidazol-1-yl)acetyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-ethyl-2-methyl-1H-indol-5-yl)-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
2,6-dimethyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]quinoline
methyl 4-({4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}amino)benzoate
N-[(5-chloro-2-methoxyphenyl)methyl]-6-(2-hydroxyethyl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-benzyl-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(cyclopropylmethyl)benzamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]oxy}benzamide
8-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-({2-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
{1-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]cyclopropyl}methanol
N-(3-hydroxypropyl)-1-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
3-[(2,5-dihydroxy-2-methylpentyl)carbamoyl]benzoic acid
1-(2,3-dimethylquinoxalin-6-yl)-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
1-(2,5-dimethylphenyl)-3-methyl-5-(1H-pyrazol-1-ylmethyl)-1H-1,2,4-triazole
2-({[(3R,4R)-4-(hydroxymethyl)-1-(4-methylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-[2-(4-fluorophenyl)ethyl]-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1,3-thiazol-2-yl)piperidine-4-carboxamide
2-methoxy-N-(1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(3S,4R)-1-[2-(4-acetylphenoxy)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
3-(3-methylthiophene-2-carbonyl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
(3S)-N-tert-butyl-2-(4-methylpiperazine-1-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-{1-[3-(azetidine-1-carbonyl)benzenesulfonyl]pyrrolidin-3-yl}piperidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-6-methyl-2-phenylpyrimidin-4-amine
N-{[3-(2-methoxyethoxy)phenyl]methyl}spiro[2.2]pentane-1-carboxamide
5-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]thiophene-2-carboxylic acid
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-2,5-dihydro-1H-pyrrole
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,6-dimethyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
(1-methanesulfonylpropan-2-yl)({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-{1-oxaspiro[4.5]decan-3-yl}urea
2-methyl-3-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
1-(2-chlorophenyl)-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2,5-dimethyl-1H-pyrrole
N3-methyl-1-(3-methylbutyl)-N5-[(2-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)(piperidin-4-ylmethyl)amine
N-[2-(4-methoxyphenyl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
N-cyclohexyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
2-[2-(dimethylamino)ethyl]-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-{[(2S,5R)-5-[(4-methylpiperazin-1-yl)methyl]oxolan-2-yl]methyl}phenyl)methyl]propanamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-(morpholine-4-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
1-(3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}phenyl)pyrrolidin-2-one
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-(thiophene-2-sulfonamido)acetamide