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1-methyl-3-phenyl-4-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[(2S,4S)-4-fluoro-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-2-yl]methyl}cyclobutanecarboxamide
5-(1,3-benzoxazol-2-yl)isoquinoline
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
N-[(3S,4R)-1-(2-hydroxypyridine-3-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
N-[(3S,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(benzyloxy)-1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
(but-2-yn-1-yl)(furan-2-ylmethyl){[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-({1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-3-phenylpyrazolo[1,5-a]pyrimidine
4-[1-(5-ethyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]pyridine
1-(2-methyl-1-benzofuran-7-carbonyl)-4-(2-phenoxyethyl)piperazine
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
N-[(3-fluorophenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)aniline
N-(3-ethoxypropyl)-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-butyl-4-hydroxy-2-(4-methylphenyl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
1-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-(2-methyl-1H-imidazol-1-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
(4aR,7aS)-1-acetyl-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopropyl-8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(3-fluorophenyl)-6,6-dimethyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(methylsulfanyl)pyridine
[3-(2-methoxyethyl)-1-(5-methyl-1,3,4-thiadiazol-2-yl)piperidin-3-yl]methanol
ethyl 4-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}piperidine-1-carboxylate
2-(1-{1-[4-(furan-2-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
N,3-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
2-{[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
N,4,6-trimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(4-cyanophenyl)-N-ethylpyridine-4-carboxamide
3,3,3-trifluoro-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]propan-1-one
1'-(oxane-4-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[(3R,4S)-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-(2-methoxyphenyl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
4-[({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}amino)methyl]-1,3-thiazol-2-amine
ethyl 2-(2-{5-[(pyridin-2-ylmethyl)carbamoyl]thiophen-2-yl}pyrrolidin-1-yl)acetate
3-[1-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-ethyl-N,3-dimethyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrazole-4-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[(4-phenylmorpholin-2-yl)methyl]propanamide
8-[2-(azepan-1-yl)acetyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}-N-cyclopropyl-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-methyl-2-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
2-ethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
7-(2-hydroxyethyl)-2-(pyridin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyridine
methyl 1-[2-hydroxy-3-(4-{[(oxan-4-yl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid