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4,6-dimethyl-N-[3-(pyridin-3-yloxy)propyl]pyrimidin-2-amine
N,N-diethyl-2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
2-(dimethylamino)-2-(2-methylphenyl)-N-[2-(propan-2-ylsulfanyl)ethyl]acetamide
10-methoxy-5-(1,3-thiazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-[5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pentyl]morpholine
(2S,4S)-4-(4-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxylic acid
9-methoxy-7-(4-methylphenyl)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(4-{1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}phenyl)methyl]-4-methylpiperazine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}propanamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-methylazepane-2-carboxamide
2-{4-[4-(dimethylamino)benzenecarbothioyl]piperazin-1-yl}-N-ethylpyridine-3-carboxamide
1-[(1S,5R)-6-[4-(difluoromethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-methoxy-6-{[8-methoxy-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
6-chloro-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
2-(3,3-diphenylpiperidin-1-yl)acetamide
1-[1'-(2,6-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-[(3-chlorophenyl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
2-(4-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
2-(1-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
2-({3-[2-(4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperazin-1-yl)ethoxy]phenyl}methyl)-2-azabicyclo[2.2.1]heptane
4-chloro-1-methyl-3-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}-1H-indazole
6-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
2-(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)ethan-1-amine
4-[(4-methoxy-3-methylphenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[2-(methylsulfanyl)benzoyl]piperidine
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
2-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
4-(2-oxo-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethoxybenzamide
6-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-3-carbonitrile
2-amino-1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
5-{[4-(6-chloropyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-(ethylsulfanyl)pyrimidine
1-{2-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-cyclohexyl-2-(2-fluorobenzoyl)-2,7-diazaspiro[4.5]decan-6-one
5-[2-(methylsulfanyl)phenoxymethyl]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
6-(cyclobutylamino)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
N,7,8-trimethyl-N-[1-(pyridin-2-yl)propan-2-yl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-3,4-dimethoxy-N-(pyridin-4-ylmethyl)benzamide
1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(4-fluorophenyl)methyl]-1-methyl-5-(4-methylpiperazin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-acetyl-8-[(3-fluoro-2-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
6-({[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]amino}methyl)-2-methylpyrimidin-4-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)butanamide
3-[3-(3-carboxyphenyl)piperidine-1-carbonyl]-5-methoxybenzoic acid
2-{4-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide