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1-(3-chlorobenzoyl)-N-(4-fluorophenyl)piperidin-3-amine
1-[1-(propan-2-yl)piperidine-3-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3aR,6aR)-2-(2-methoxyethyl)-5-(1-phenylcyclopropanecarbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-2-phenylpyrimidin-4-ol
2-amino-4-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}quinazoline-6-carboxylic acid
3-{[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
(1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[(2-methylphenyl)methyl]piperidin-3-yl)methanol
3-methoxy-N-[1-(4-methoxy-3-methylphenyl)ethyl]-2,2-dimethylpropanamide
1'-(2-chloro-4-fluorobenzoyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(2,6-dimethoxypyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(pyridine-2-carbonyl)-1,4-diazepan-2-one
1-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}imidazolidin-2-one
8-(2-methoxyacetyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(2-fluorophenyl)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3aR,6aS)-2-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-octahydropyrrolo[3,4-c]pyrrole
N-(3,5-dimethoxyphenyl)-3-[1-(1H-imidazole-2-carbonyl)piperidin-3-yl]propanamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[4-methyl-3-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-{1-[(3,4-dimethoxyphenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-(oxolan-2-ylmethyl)urea
4-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[3-(1H-pyrazol-4-yl)benzoyl]-1,4-diazepan-5-one
N-(9H-fluoren-9-yl)-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxylic acid
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]propanoic acid
1-methyl-N-[1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]piperidine-4-carboxamide
2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-4,6-dimethoxypyrimidine
1-(1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-4-(4-fluorophenyl)piperazine
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
2-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)-N-[2-(3-fluorophenyl)ethyl]acetamide
N,4-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
[(2,3-difluoro-6-methoxyphenyl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
7-cyclobutanecarbonyl-N,N-dimethyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(benzyloxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-[(8-methoxyquinolin-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[1-(4-cyclobutyl-6-methylpyrimidin-2-yl)pyrrolidin-3-yl]acetamide
3-{[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}-1-phenylpropan-1-ol
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
(4S)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}-4-(pyrrolidin-1-yl)pentan-1-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[1-(methoxymethyl)cyclopentyl]methyl}acetamide
1-(3-chloro-4-methoxyphenyl)-3-(3-methoxypropyl)-3-(1-methylpiperidin-4-yl)urea
(furan-3-ylmethyl)(methyl){[(2R,5S)-5-[(2-methylpyridin-4-yl)methyl]oxolan-2-yl]methyl}amine
(3S,4S)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
3-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methoxy)pyridine-2-carbonitrile
2-methyl-4-phenyl-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]quinoxaline-6-carboxamide
(2E)-N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(pyridin-2-yl)prop-2-enamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
methyl 3-(2-chloro-6-fluorobenzamido)-6-[(2-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate