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3-{4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}-N-(pyridin-3-yl)propanamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2,3-dimethylphenoxy)ethan-1-one
4-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
1-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)propan-1-one
7-(1,3-benzothiazol-2-yl)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[4-(3-hydroxypropyl)-1H-1,2,3-triazol-1-yl]-N-(2-phenylethyl)piperidine-1-carboxamide
3-ethoxy-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
5-acetyl-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methoxy-4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
(3aR,7aS)-2-[2-methoxy-5-(1,2-oxazol-5-yl)benzenesulfonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-(3-{[1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
2-(dimethylamino)-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-2-(3-methylphenyl)acetamide
5-[({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
8-(3-ethoxyphenyl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-methyl-5-propyl-4-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidine
N,2-dimethyl-4-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidine-5-carboxamide
2-(3-fluorophenyl)-1-[(4-methanesulfonylphenyl)methyl]piperidine
5-oxo-1-[4-(propan-2-yl)phenyl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidine-3-carboxamide
(4S,4aS,8aS)-4-hydroxy-N,N-dimethyl-4-phenyl-decahydroquinoline-1-sulfonamide
N,N-dimethyl-2-{methyl[(1-phenyl-1H-pyrazol-5-yl)methyl]amino}propanamide
6-(4-fluorophenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[4-(trifluoromethyl)phenyl]urea
5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-imidazole-4-carboxylic acid
1,6-dimethyl-3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
1-(4-cyclohexylpiperazin-1-yl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-(3-methylcinnolin-5-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
5-methanesulfonyl-N-(2-phenylethyl)-4-(piperidin-3-yl)pyrimidin-2-amine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
6-fluoro-4-(1,3-thiazol-5-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(3R,4R)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carboxamide
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-(1,3-benzothiazol-2-ylmethyl)-5-(1-benzyl-4-hydroxypiperidin-4-yl)-1-benzofuran-2-carboxamide
methyl 3-benzamido-5-{[(3-methylphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(4-methoxyphenyl)-5-methyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperazin-2-one
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-3-(furan-2-yl)propan-1-one
4-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-oxobutane-1-sulfonamide
2-methoxy-6-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}phenol
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(3-methylpyridin-2-yl)piperazine
7-phenyl-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N,2,6-trimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}pyridine-4-carboxamide
9-(3-phenoxybenzoyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1R,2R)-2-{[(6-ethylpyrimidin-4-yl)amino]methyl}-1-methylcyclohexan-1-ol
2-[3-(1-phenylcyclopropyl)-5-(4-propylpyrimidin-5-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-(4-methylpiperazin-1-yl)propanamide
(5S,9aS,9bS)-5-[(E)-2-(furan-2-yl)ethenyl]-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-propylpyridine-4-carboxamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide