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1-({1-[6-(cycloheptylamino)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-[2-(methylsulfanyl)phenyl]acetamide
2-amino-4-(2-ethylpyrimidin-5-yl)-7-hydroxy-5H,6H-benzo[h]quinoline-3-carbonitrile
(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-[(cyclobutylamino)methyl]-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
6-fluoro-2-oxo-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-cyclopropyl-9-(2-methoxyethyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
4-(5-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}furan-2-yl)-2-methylbut-3-yn-2-ol
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-phenoxyethan-1-one
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-2-[2-(methylsulfanyl)benzoyl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(4-methylphenyl)-4-(6-methylpyridine-3-carbonyl)piperazin-2-one
2-{5-[1-(2,4-difluorophenoxy)ethyl]-3-methyl-1H-1,2,4-triazol-1-yl}-6-methylpyridine
6-(azepan-1-yl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methylpyridine-3-carboxamide
methyl (2S)-1-{2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)pyridine-3-carbonyl}pyrrolidine-2-carboxylate
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-(2-methoxyacetyl)piperidine-4-carboxamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
1-{4-[4-(dimethylamino)azepane-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-methyl-6-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyrimidin-4-ol
1-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-(3-methylthiophen-2-yl)-1H-1,2,3-triazole
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)amino]-N,N-dimethylethane-1-sulfonamide
4-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-3-(3-methylphenoxymethyl)piperidine
2-(carbamoylamino)-N-[(3R,4S)-1-[(2-chlorophenyl)methyl]-4-cyclopropylpyrrolidin-3-yl]acetamide
ethyl 1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxylate
N-[(2-methoxyphenyl)methyl]-2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}acetamide
N-{1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1-methylpyrrolidin-3-yl)pyridin-2-amine
N-{2-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]ethyl}-4-fluorobenzamide
2-{3-[(3-chlorophenyl)methyl]-5-[(2-oxo-1,2-dihydropyridin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-chloro-N-[2-(pyridin-4-yl)ethyl]-5-(trifluoromethyl)benzamide
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3-[2-(2-methylpropanesulfonyl)ethyl]urea
1-(2-methoxy-6-methylbenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
5-methyl-4-[3-methyl-1-(4-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(prop-2-en-1-yl)-1H-pyrazole
4-[5-(3,5-dimethyl-1H-pyrazol-4-yl)furan-2-carbonyl]morpholine
5-fluoro-2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3-azaspiro[5.5]undecan-9-amine
4-methyl-6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-2-amine
N-{2-[4-(2-chloro-6-fluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-3-methylpyridin-4-amine
7-(3,5-dimethoxybenzoyl)-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane
methyl 4-({4-[2-(2-fluorophenyl)-1-(N-methyl-1-thiophen-3-ylformamido)ethyl]piperidin-1-yl}methyl)benzoate
2-({4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}sulfanyl)ethan-1-ol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazole-3-carboxamide
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{4-[(3-methoxyphenyl)methyl]morpholin-3-yl}acetamide
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methoxyphenol
N-(3,3-diphenylpropyl)-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane