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(3R,4R)-1-(5-propyl-1,2,4-oxadiazol-3-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
2-ethyl-4-phenyl-9-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane
6,7-dimethyl-2-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
methyl 3-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{1-[2-(4-benzyl-2-oxopyrrolidin-1-yl)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-[3-(dimethylamino)-1-phenylpropyl]-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{4-[(6-chloropyridin-3-yl)methyl]piperazine-1-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
3-chloro-5-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
2-(furan-2-yl)-5-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}pyrimidine
{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}(propyl)(pyridin-3-ylmethyl)amine
2-[5-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)furan-2-yl]benzonitrile
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(piperidin-1-yl)acetamide
1-[(3,5-dichloropyridin-4-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
[1-(3-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propyl)piperidin-2-yl]methanol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]pyrimidine
7-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-tert-butyl-1,2,4-oxadiazole
[(5-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}thiophen-3-yl)methyl]dimethylamine
5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-2-(3-phenoxyphenyl)-1,3-oxazole
1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
4-ethyl-3-({1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-benzyl-1-(3,4-dimethylbenzoyl)-3-ethyl-1,4-diazepan-5-one
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
methyl (2S,4R)-1-{[4-(propan-2-yl)phenyl]methyl}-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
3-{2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1H-pyrazol-5-amine
(3aS,6aS)-2-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[1-(7-fluoro-2-methylquinoline-4-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
5-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}-1H-indole
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
(2S,4S)-4-(4-{[(tert-butylcarbamoyl)(methyl)amino]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxylic acid
6-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
6-methyl-5-{5-[4-(piperidin-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
(4aS,8aR)-6-(5-fluoro-2-methylbenzoyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
2-(dimethylamino)-7-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[3-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)phenoxy]ethan-1-ol
2-methyl-5-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
(3R,4S)-1-[4-methoxy-3-(morpholin-4-yl)benzoyl]-3,4-dimethylpiperidin-4-ol
3-(4-methyl-1,3-thiazol-5-yl)-1-(thiomorpholin-4-yl)propan-1-one
N-[(4-fluorophenyl)methyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-cyclopropyl-3-(2-fluorophenyl)-N-[(3-hydroxyphenyl)methyl]-1H-pyrazole-4-carboxamide
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-4-(2-propylpyrrolidine-1-carbonyl)-2,3-dihydro-1H-isoindol-1-one
1-(3-chloropyridin-2-yl)-4-(1H-imidazol-4-ylmethyl)piperazine
1-[2-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
1-(2-methylphenyl)-4-[1-(thiophene-3-carbonyl)piperidin-3-yl]piperazine
3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-[1-(pyrimidin-4-yl)ethyl]urea
N-{3-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)carbamoyl)methoxy]phenyl}propanamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine