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3-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-{2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
methyl[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](1,2-oxazol-3-ylmethyl)amine
(3S,4R)-4-(2-methylphenyl)-1-(6-methylpyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
3-fluoro-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]benzonitrile
N-(6-methylpyridin-3-yl)-1-(5-methylpyridine-3-carbonyl)piperazine-2-carboxamide
ethyl 2-{[2-(4-cyclopentylpiperazine-1-carbonyl)phenyl]amino}acetate
(4aS,8aR)-N-cyclohexyl-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
5-{2-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-cyclopentyl-4-(methylamino)-N-propylbenzamide
10-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
1-{2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
(2R,3S,6R)-3-(2-methoxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]ethan-1-one
1,3-dimethyl-4-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole
1-({1-[6-(3-hydroxyazetidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-[4-(cyclohex-3-en-1-ylmethyl)piperazin-1-yl]quinazoline
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-(2-methylphenoxy)acetamide
1-[(2-aminopyrimidin-5-yl)methyl]-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
4-(2H-1,3-benzodioxol-5-yloxy)-1-(2-cyclopropylacetyl)piperidine-4-carboxylic acid
N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[(5-methylthiophen-2-yl)methyl]pyridin-2-amine
4-chloro-2-fluoro-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
2-(3-methoxyphenoxymethyl)-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
2,6-difluoro-4-methoxy-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
N-[1-(2,4-difluorophenyl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(2-aminoethyl)-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
[3-(2-methoxyethyl)-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl]methanol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1'-(3-hydroxy-2-methylbenzoyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
2-(dimethyl-1,3-thiazol-5-yl)-1-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}ethan-1-one
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
5-(1H-1,3-benzodiazole-5-carbonyl)-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{2-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-(1-cycloheptylpiperidin-3-yl)-3,5-dimethyl-1H-pyrrole-2-carboxamide
N-{1-[1-(3-fluoropropyl)-1,2,5,6-tetrahydropyridin-3-yl]propan-2-yl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]benzamide
8-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-2-yl]pyridine
3-(2-ethyl-1H-imidazol-1-yl)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]propanamide
2-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}sulfonyl)benzonitrile
1-(2,3-dimethylquinoxalin-6-yl)-3-[(2-propyl-1,3-thiazol-4-yl)methyl]urea
N-{2-ethyl-4-[3-(1H-pyrazol-1-yl)phenyl]phenyl}acetamide
3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(benzyloxy)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one