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[(1-cyclohexylpiperidin-3-yl)methyl]({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(pyridin-3-ylmethyl)amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-(1H-pyrazol-1-yl)butanamide
4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-1-(1H-indazol-5-yl)piperazin-2-one
N-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
2-(3-oxopiperazin-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
7-(3-chlorophenyl)-4-(1-methyl-1H-pyrazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 4-oxo-5-phenoxy-1-[(1-propyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3-carboxylate
N-[(3-hydroxyphenyl)methyl]-N-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
methyl[4-(morpholin-4-yl)butyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
(4aS,8aR)-6-[(3-methyl-1-benzofuran-2-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine-4-carboxylic acid
3-methyl-4-({3-[3-(pyridin-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
(1S,5R)-6-[(3-chloro-4-fluorophenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-(benzyloxy)-8-(2,6-dimethoxypyridine-3-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
N-[(2,5-dimethylphenyl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
1-(2-methylpyridin-4-yl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,4-diazepane
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(3aS,6aS)-1-(4-phenoxybutyl)-octahydropyrrolo[2,3-c]pyrrole
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methyl-1H-indazole-3-carboxamide
2-chloro-N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
4-methyl-2-[4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
1-(5-chloropyridin-2-yl)-4-(2-methyloxane-2-carbonyl)piperazine
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-imidazole-2-carboxamide
8-fluoro-2-({[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amino}methyl)quinolin-4-ol
2-[2-(dimethylamino)ethyl]-8-[2-(1H-1,2,3,4-tetrazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-cyclopentyl-N-(3-methylbutyl)-4-oxo-5-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[(3S,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-ylmethyl}acetamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(cyclohex-1-en-1-yl)ethyl]acetamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-{[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}-N-(2-hydroxyethyl)pyridine-2-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}propan-1-one
4-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-ethyl-5-(4-methyl-2-phenylpiperazine-1-carbonyl)pyrimidine
2-amino-1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
N,N-dimethyl-5-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]-1,3-thiazol-2-amine
4-[(2,4-difluorophenyl)methyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[(3R,4R)-1-[(5-cyano-1H-pyrrol-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
3-{5-[3-(piperazin-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
(2-{2-[1-(3-ethoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-(furan-2-yl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)azepane
4-({2-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-3-(1,2-oxazinan-2-yl)propanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(4-methylpiperazin-1-yl)propyl]acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
(1R,5S,8R)-8-(dimethylamino)-N-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide