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1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-phenylpropyl)pyrrolidin-3-yl]methanol
8-[(5-carboxy-2-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
N-(2,3-dihydro-1H-inden-2-yl)-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
methyl 4-{[({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]methyl}benzoate
2-(2-{1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-(1-ethylcyclopropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-[3-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-(1-hydroxy-2-methylpropan-2-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-(6-methoxypyridin-3-yl)pyridine-3-carboxylate
N,2-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
2-(4-methylpentyl)-4-(pyridin-4-ylmethyl)morpholine
N-[1-(4-methanesulfonylphenyl)propyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[4-(methylsulfanyl)phenyl]methyl}-4-oxo-N-(prop-2-en-1-yl)pentanamide
2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]acetamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2-phenylbenzoyl)piperidine
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
N-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)acetamide
3-[1-(3-ethoxypropyl)-1H-imidazol-2-yl]-1-methyl-1,2-dihydroquinolin-2-one
5-phenyl-N-[1-(pyridin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(4H-1,2,4-triazol-4-yl)piperidine
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-cyclobutanecarbonyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(4aR,8aR)-7-(2-chloro-5-fluorobenzoyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
(1S,5R)-6-(2-methoxyethyl)-3-(5-phenyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethylamino)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2,3-dihydro-1H-indene-2-carboxamide
2-[4-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-(4-chlorophenoxy)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
5-(1H-pyrazol-3-ylmethyl)-2-[3-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
methyl 4-methoxy-3-[2-(propan-2-yl)-1H-imidazol-1-yl]benzoate
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-{[(2-methoxyethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-(2-methyl-6-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}pyrimidin-4-yl)ethan-1-amine
4-(2-ethoxyethyl)-N-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}piperazine-1-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-{[3-(morpholin-4-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-butyl-4-{[(2-methoxyphenyl)methyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
N-(4-methoxy-2-methylphenyl)-3-[1-(3-phenylpropanoyl)piperidin-3-yl]propanamide
{2-oxo-2-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}urea
2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[4-(4-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
N-(2,1,3-benzoxadiazol-4-ylmethyl)-6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
dimethyl({2-[4-(6-methylquinoline-4-carbonyl)morpholin-2-yl]ethyl})amine
3-cyclohexyl-N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-[3-(1H-indol-1-yl)propyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
N-ethyl-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine