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3-(2-aminoethyl)-5-(furan-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
N-[(2-ethylpyrimidin-5-yl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
8-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl][4-(trifluoromethyl)phenyl]methanol
4,6-dimethyl-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}quinoline
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
4-({[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}amino)-2-methoxypyridine-3-carbonitrile
(3aS,6aR)-5-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-(2,6-difluoro-3-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-cyclopropyl-9-(2-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,7S)-N-methyl-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-ethyl-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-methyl-1H-pyrazole-4-carboxamide
6-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-amino-4-[4-ethoxy-3-(hydroxymethyl)phenyl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
9-methoxy-7-(4-methoxyphenyl)-4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]pyrazin-2-ol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-(2-ethylphenyl)-3-[(thiolan-3-yl)amino]propanamide
N-cyclopropyl-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-ol
4-(7-hydroxyquinolin-3-yl)-5,7-dimethoxy-1,2,3,4-tetrahydroquinolin-2-one
N-[2-methyl-5-({[1-(oxolan-2-ylmethyl)piperidin-4-yl]carbamoyl}amino)phenyl]propanamide
1-[2-(morpholin-4-yl)ethyl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[(1-benzylpiperidin-4-yl)amino]-N-(2-methylphenyl)propanamide
5-chloro-N-{1,9-dioxaspiro[5.5]undecan-4-yl}thiophene-2-carboxamide
2-[2-(dimethylamino)ethyl]-9-[(4-fluoro-3-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[1-(3-chloro-4-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
(1R,9S)-5-amino-3-(5-methoxy-1H-indazol-3-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
4-(furan-3-ylmethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(1R,2S)-N1-butyl-N2-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]cyclohexane-1,2-dicarboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]propanamide
N-{2-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
5-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-methylpyrrolidin-2-one
(3S,4S)-1-(4-methyl-1,3-oxazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-{4-[3-({[(2-chloro-4-fluorophenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
methyl 4-(5-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-(3,4-dichlorophenyl)-4-(3-methylpyrazin-2-yl)morpholine
N-[(2S,4R,6R)-2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-6-(propan-2-yl)oxan-4-yl]acetamide
6-{4-[(3-ethenylphenyl)methyl]piperazin-1-yl}-N,N-dimethylpyrazine-2-carboxamide
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})(pyrrolidin-3-ylmethyl)amine
3-[(1H-imidazol-2-ylmethyl)(prop-2-en-1-yl)amino]-3-methyl-1λ6-thiolane-1,1-dione
2-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylbenzamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
2-[(1S,5R)-6-[(2,3-dichlorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-(2-methoxyethyl)-1-(2-methyl-5-sulfamoylphenyl)-3-(1,3-thiazol-2-ylmethyl)urea
8-[1-(cyclopropylmethyl)-7-oxoazepan-4-yl]-2-(diethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-cyclobutyl-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1,3,4-oxadiazol-2-amine
2-[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]-5-fluoro-1H-1,3-benzodiazole
2-{4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}ethan-1-ol