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N-ethyl-6-methyl-N-[2-(morpholin-4-yl)ethyl]pyridine-2-carboxamide
1-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-fluoro-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-sulfamoylbenzamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
1-(4-ethylpiperazin-1-yl)-3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}propan-1-one
4-(4-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
N-(2,4-dimethylphenyl)-3-({6-methylpyrazolo[1,5-a]pyrimidin-3-yl}formamido)propanamide
1-[3-(3-chlorophenoxy)azetidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
1-(2,3-dimethylquinoxaline-6-carbonyl)azepan-4-amine
3-[(methylsulfanyl)methyl]-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidine
6-(2-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(7R,8aS)-7-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-(3-hydroxy-3-methylbutyl)-N-[(2S)-1-hydroxypropan-2-yl]benzamide
2-(4-hydroxy-3,3-dimethylbutyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-(2,4-dimethylphenyl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
4-[(1-{2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)oxy]pyridine
1-ethyl-4-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
methyl 3-(1-benzofuran-2-ylmethyl)-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(4-cyclopentylpyrimidin-2-yl)amino]-N-methylpentanamide
6-methoxy-4-[4-(2-methoxyacetyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}dimethylamine
(3S,5R)-1-(cyclopropylmethyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-[2-(ethanesulfonyl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(3-fluorophenyl)methyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
[(2S,4R)-4-(dimethylamino)-1-[(6-methoxypyridin-3-yl)methyl]pyrrolidin-2-yl]methanol
2,3-dimethoxy-N-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methyl}benzamide
5-[(4-fluorophenyl)methyl]-5-[1-(pyrrolidine-1-sulfonyl)piperidin-4-yl]imidazolidine-2,4-dione
8-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-{2-[(4-ethylpiperazin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-(2-methoxyethoxy)ethan-1-one
2-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-6-(trifluoromethyl)pyridine-3-carboxamide
(3S)-N,N-dimethyl-1-(2-methyl-4-phenylpyridine-3-carbonyl)azepan-3-amine
(3R,4R)-4-ethyl-1-(isoquinolin-1-yl)piperidine-3,4-diol
N-(dimethyl-1,2-oxazol-4-yl)-4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
2-(4-oxo-1,4-dihydroquinolin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
3-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(furan-2-ylmethyl)(methyl){[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
11-methyl-5-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
2-methyl-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrazine
5-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(4-ethylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3S)-3-ethylmorpholin-4-yl]-4-(1H-pyrazol-1-yl)butan-1-one
2-hydroxy-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
3-(3-fluorophenoxymethyl)-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
(3S)-4-(6,7-diethoxy-3-methyl-1-benzofuran-2-carbonyl)-3-ethylmorpholine
3-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-6-methoxy-1H-indazole
4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide