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5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}piperidin-2-one
4-{5-[(2,5-dimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1,5-dimethyl-1H-pyrazole
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
6-(1-{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-2-methyl-3,4-dihydropyrimidin-4-one
2-benzyl-8-[2-(phenylsulfanyl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
2-(1-benzothiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(2S,4S)-N-ethyl-4-[2-(propylsulfanyl)acetamido]-1-(1H-pyrrole-3-carbonyl)pyrrolidine-2-carboxamide
6-cyclopentyl-1-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(5S,9aS,9bS)-5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[1-(6-amino-2-methylpyrimidin-4-yl)piperidin-4-yl]-1,3-oxazolidin-2-one
1-{3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
5-(1-benzofuran-2-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
2-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
6-[(diethylamino)methyl]-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[(3-methylpiperazin-1-yl)sulfonyl]-N-[2-(pyrazin-2-yl)ethyl]benzamide
1-(isoquinolin-1-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-methyl-4-{3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
2-(diethylamino)-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-(2,7,8-trimethylquinoline-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
ethyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
1-methyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
(3aS,6aR)-5-(5-methyl-1,3-benzoxazol-2-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[2-(5-acetylthiophen-3-yl)acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(thiophen-2-yl)ethyl]-1-{2-[(3,4,5-trimethoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-chloro-6-[3-(3-methoxypropyl)piperidin-1-yl]pyridine-2-carboxylic acid
[(1-cyclopentylpiperidin-4-yl)methyl]({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})(pyridin-3-ylmethyl)amine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
methyl 4-{[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
(2S)-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamidopropanamide
2-ethoxy-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
4-ethyl-1-methyl-3-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1,2-oxazolidin-2-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)propanamide
4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-(4-chlorophenyl)-5-(2-phenoxyethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-(2-amino-4-{[3-(2,3-dihydro-1H-indol-1-yl)propyl]amino}-6-methylpyrimidin-5-yl)propanoic acid
1-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}pent-4-en-1-one
N3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-N1,N1-dimethylpiperidine-1,3-dicarboxamide
1-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}-4-phenylbutan-1-one
1-[(3-chlorophenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
8-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-(1-cycloheptylpiperidin-3-yl)-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazin-2-one
9-methoxy-4-[(3-methoxyphenyl)methyl]-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-ethyl-N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-ethyl-3-(propan-2-yl)-N-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]piperidin-3-ol