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2-{2-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(pyridin-3-yl)-3-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}propanamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-(1H-imidazol-2-ylmethyl)propanamide
6-methyl-3-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[4-({3-[3-(6-methylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}methyl)thiophen-2-yl]ethan-1-one
4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2-(3-phenylpropyl)morpholine
1-(1-{1-[1-(trifluoromethyl)cyclopropanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)cyclopentan-1-ol
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-1-propyl-1H-pyrazole-5-carboxamide
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-3,5-dimethyl-1-benzofuran-2-carboxamide
4-[(4-methoxyphenyl)methyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-5-one
6-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
6-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[(3R,5S)-1-[(2-aminopyridin-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
1-[(3S,4R)-1-(4-methoxyquinoline-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[2-(piperidin-1-ylmethyl)phenyl]urea
3-{1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
4-({4-[1-(dimethylamino)ethyl]piperidin-1-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
2-{[(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-3-yl)oxy]methyl}pyridine
1-(oxan-4-yl)-4-(1H-pyrazole-3-carbonyl)-1,4-diazepan-6-ol
2-methyl-4-[4-(oxan-4-yl)piperazin-1-yl]-6-(piperidin-3-yl)pyrimidine
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
5-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
6-cyclobutyl-2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-{2-[2-(3-ethyl-1H-pyrazol-5-yl)-1H-imidazol-1-yl]ethyl}morpholine
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylbenzamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-[4-(methylsulfanyl)phenyl]acetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(pyridin-2-ylsulfanyl)acetamide
4-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-[3-(trifluoromethoxy)phenyl]urea
3-[({[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}amino)methyl]piperidin-3-ol
5-[4-(aminomethyl)piperidin-1-yl]-2-(cyclobutylmethyl)-2,3-dihydropyridazin-3-one
5-(3,4-dimethoxyphenyl)-3-[4-(thiomorpholin-4-yl)piperidin-1-yl]-1,2,4-triazine
1-[3-(3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
[(3S,5R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
N,N-dimethyl-6-oxo-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-sulfonamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[4-(morpholin-4-yl)phenyl]acetamide
1-(4-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
N-(1-methyl-1H-pyrazol-5-yl)-2-[3-(quinolin-8-yl)-1H-indazol-1-yl]acetamide
1-methyl-4-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperazin-2-one
5-[2-(dimethylamino)propanoyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-(2-fluorophenyl)-3-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)propanamide
N-ethyl-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-amine
4-(3,4-difluorophenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
14-[2-(furan-2-yl)phenyl]-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}-1,4-diazepan-5-one
2-(4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}quinazolin-2-yl)ethan-1-amine
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
5-methyl-4-[(prop-2-en-1-yl)amino]-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide