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1-{1-[2-(4-hydroxy-2,6-dimethylpyrimidin-5-yl)acetyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(pyridin-4-yl)propan-1-one
methyl 1-[(3S,5S)-1-[(3-fluorophenyl)methyl]-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
6-[4-(thiomorpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]pyridine-2-carbonitrile
2-{5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-phenylazepane
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](1H-indol-7-ylmethyl)methylamine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(5-oxopyrrolidin-2-yl)acetamide
8-(2,6-difluorobenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(morpholin-4-yl)ethyl]-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-2-one
N-ethyl-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(2-hydroxyethyl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
(2S)-2-(methylamino)-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one
3-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-benzyl-5-[(3,4-dimethylpiperazin-1-yl)methyl]pyrimidin-2-amine
(5S,9aS,9bS)-5-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[2-(pyridin-2-yl)ethyl]benzamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-4-propyl-1,2,3-thiadiazole-5-carboxamide
2-{5-[2-(2,3-dihydro-1H-inden-5-yloxy)propan-2-yl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[(1S)-1-phenylpropyl]piperidine-1-carboxamide
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide
3-{[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
(1R,3S)-3-(2-aminoethoxy)-7-(1-benzofuran-2-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
7-[(2,3-dimethoxyphenyl)methyl]-2-(1H-imidazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[5-(2-methyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[(oxolan-3-yl)amino]piperidin-1-yl}phenyl)acetamide
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]propanamide
2-amino-4-(furan-3-yl)-6-(1H-indol-3-yl)pyridine-3-carbonitrile
(3S,4S)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2-fluoro-4-methylbenzoyl)piperidine
1-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-methylurea
(1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-yl)methanamine
5-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl}-4-methylpiperazine
6-fluoro-2-{[(6-hydroxy-6-methylheptan-2-yl)amino]methyl}quinolin-4-ol
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
ethyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
1-(5-hydroxypyrazine-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
4-benzyl-3-ethyl-1-(1-ethylpiperidin-4-yl)-1,4-diazepan-5-one
2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxylic acid
1-(3-chloro-2-fluorophenyl)-5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-methyl-1H-1,2,4-triazole
4-(4-methyl-1H-pyrazol-1-yl)-1-(2-phenoxyacetyl)piperidine-4-carboxylic acid
1-[(2R,3R)-3-[ethyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
methyl[(3-{[1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](thiophen-3-ylmethyl)amine
ethyl 5-(5-methyl-1H-pyrazole-3-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate